SCHEMBL7170677

SCHEMBL7170677

NN(c1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.41
CES2 O00748 1/20 0.41
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
IKBKB O14920 1/20 0.36
TACR1 P25103 2/20 0.36
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
PTPN5 P54829 1/20 0.33
P2RX1 P51575 1/20 0.33
TDO2 P48775 1/20 0.33
ADRB1 P08588 1/20 0.33
GAA P10253 1/20 0.33
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL440959 0.76 CES2 (0.58) IDO1CES2ITGB3ITGAVTSHR
SCHEMBL12964480 0.76 CES2 (0.42) IDO1CES2ITGB3ITGAVTACR1
SCHEMBL5537293 0.76 CES2 (0.42) IDO1CES2ITGB3ITGAVTACR1
SCHEMBL7694014 0.74 TACR1 (0.43) IDO1CES2TACR1TSHRP2RX1
SCHEMBL657091 0.74 TACR1 (0.43) IDO1CES2TACR1P2RX1
SCHEMBL5535744 0.74 CES2 (0.41) IDO1CES2ITGB3ITGAVTACR1
SCHEMBL15800804 0.72 TSHR (0.48) IDO1CES2TSHRMAPK1TDO2
SCHEMBL12937113 0.72 CES2 (0.39) IDO1CES2TACR1TSHRMAPK1
SCHEMBL16345980 0.70 CES2 (0.48) IDO1CES2ITGB3ITGAVTACR1
SCHEMBL15323725 0.70 ALDH1A1 (0.43) IDO1CES2ITGB3ITGAVTACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003007955-A2 BIPHENYL APURINIC/APYRIMIDINIC SITE ENDONUCLEASE INHIBITORS TO TREAT CANCER CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2003-01-30 WO claimed