SCHEMBL7174972

SCHEMBL7174972

Cc1ccc(NC(=S)N(CCc2cncn2Cc2ccc([N+](=O)[O-])cc2)Cc2cccc(Cl)c2Cl)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.43
MAPT P10636 7/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
HTT P42858 4/20 0.43
GAA P10253 1/20 0.43
FNTA P49354 2/20 0.41
FNTB P49356 2/20 0.41
PGGT1B P53609 2/20 0.41
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.41
NPSR1 Q6W5P4 4/20 0.40
POLB P06746 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTR1E P28566 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083742 0.90 MMP1 (0.44) ALDH1A1MAPTSMN1; SMN2HTTFNTA
SCHEMBL7077725 0.90 YES1 (0.41) ALDH1A1MAPTSMN1; SMN2HTTGAA
SCHEMBL7076590 0.88 CYP11B1 (0.43) ALDH1A1MAPTSMN1; SMN2HTTFNTA
SCHEMBL7078782 0.81 ALDH1A1 (0.45) ALDH1A1MAPTSMN1; SMN2HTTGAA
SCHEMBL7178460 0.79 FNTA (0.46) ALDH1A1MAPTSMN1; SMN2HTTGAA
SCHEMBL7083066 0.77 KCNH2 (0.47) ALDH1A1MAPTSMN1; SMN2HTTGAA
SCHEMBL7083275 0.76 CYP11B1 (0.46) FNTAFNTBPGGT1B
SCHEMBL8582869 0.76 FNTA (0.39) ALDH1A1FNTAFNTBPGGT1B
SCHEMBL7076893 0.76 ALDH1A1 (0.42) ALDH1A1MAPTSMN1; SMN2HTTGAA
SCHEMBL7173341 0.75 CYP11B1 (0.44) ALDH1A1MAPTSMN1; SMN2HTTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1200430-A4 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORP LTD (KR) 2003-01-22 EP disclosed
EP-1200430-A1 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORPORATION, LTD. (KR) 2002-05-02 EP disclosed
WO-2001009128-A1 THIOUREA AND ISOTHIOUREA DERIVATIVES FOR INHIBITING RAS-TRANSFORMED CELL GROWTH YUHAN CORPORATION (KR) 2001-02-08 WO disclosed