SCHEMBL7176290

SCHEMBL7176290

COC=CCc1ncccn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23037266 0.75 HSP90AA1 (0.33)
SCHEMBL23037268 0.75 HSP90AA1 (0.33)
SCHEMBL8591170 0.71 LOXL2 (0.50)
SCHEMBL6159661 0.70
SCHEMBL10746552 0.70
SCHEMBL1257944 0.70 HSP90AA1 (0.33)
SCHEMBL6429020 0.70 HSP90AA1 (0.33)
SCHEMBL1247038 0.70
SCHEMBL4588569 0.69
SCHEMBL8703080 0.68 ALDH1A1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6555676-B2 Antitumor agents CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2003-04-29 US claimed
US-20020037873-A1 Biologically active phosphotriester-type compounds CENTRE NATIONAL DE LA RECHERCH SIENTIFIQUE 2002-03-28 US claimed
US-5849905-A Biologically active phosphotriester-type nucleosides and methods for preparing same CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 1998-12-15 US claimed
US-5770725-A USES NOVEL GROUP, CHARACTERIZED BY THE PRESENCE OF-S-S-AND/OR S-C=Z (Z=O OR S) ENZYME LABILE BONDS WHICH LEADS, AFTER ENZYMATIC ACTIVATION, TO THE FORMATION OF UNSTABLE INTERMEDIATE WHICH RELEASES MONOPHOSPHATE OR MONOPHOSPHONATE CENTER NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 1998-06-23 US claimed
WO-1998011121-A1 BIOLOGICALLY ACTIVE PHOSPHOTRIESTER-TYPE COMPOUNDS CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 1998-03-19 WO claimed