SCHEMBL7182870

SCHEMBL7182870

CC(C)(NC(=O)c1c[c]cc(Nc2ccccc2)c1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 3/20 0.44
TACR3 P29371 1/20 0.40
ROCK2 O75116 2/20 0.39
ROCK1 Q13464 1/20 0.39
PPARG P37231 1/20 0.39
KCNK9 Q9NPC2 1/20 0.38
EGLN1 Q9GZT9 2/20 0.38
PHGDH O43175 1/20 0.37
MAPT P10636 2/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
CNR2 P34972 1/20 0.37
MEN1 O00255 1/20 0.36
CASP3 P42574 1/20 0.36
KMT2A Q03164 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36
SSTR4 P31391 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6530802 0.81 IMPDH2 (0.48) IMPDH2TACR3ROCK2ROCK1PPARG
SCHEMBL7592814 0.77 HDAC6 (0.43) MAPTGAAHPGDMEN1CASP3
SCHEMBL3039120 0.75 POLB (0.58) IMPDH2TACR3ROCK2ROCK1KCNK9
SCHEMBL7195286 0.74 KMT2A (0.52) MAPTGAAHPGDCNR2MEN1
SCHEMBL7674538 0.73 SIRT2 (0.51) PPARGHPGDRAB9AKMT2AHDAC1
SCHEMBL7182884 0.71 NPC1 (0.48) ROCK2ROCK1MAPTRAB9A
SCHEMBL17585366 0.70 POLB (0.53) IMPDH2TACR3ROCK2KCNK9GAA
SCHEMBL3836272 0.70 RAB9A (0.57) IMPDH2ROCK2KCNK9RAB9ACASP3
SCHEMBL94229 0.69 IMPDH2 (0.52) IMPDH2TACR3ROCK2ROCK1KCNK9
SCHEMBL3838597 0.69 IMPDH2 (0.52) IMPDH2TACR3ROCK2ROCK1EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1274676-A2 POLYCYCLIC ARYL AND HETEROARYL SUBSTITUTED 1,4-QUINONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE Pharmacia Corporation (US) 2003-01-15 EP claimed
WO-2001079155-A2 POLYCYCLIC ARYL AND HETEROARYL SUBSTITUTED 1,4-QUINONES USEFUL FOR SELECTIVE INHIBITION OF THE COAGULATION CASCADE PHARMACIA CORPORATION (US) 2001-10-25 WO claimed