SCHEMBL7185015

SCHEMBL7185015

O=C(O)C=Cc1ccc(Oc2c(-c3ccc(O)c(Cl)c3)ccc3ccccc23)cc1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 17/20 0.50
ESR2 Q92731 10/20 0.50
PTPN11 Q06124 1/20 0.45
ABCG2 Q9UNQ0 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185012 1.00 ESR1 (0.50) ESR1ESR2PTPN11ABCG2
SCHEMBL7188316 0.89 ESR1 (0.41) ESR1ESR2ABCG2
SCHEMBL7188311 0.89 ESR1 (0.41) ESR1ESR2ABCG2
SCHEMBL7182554 0.87 ESR1 (0.52) ESR1ESR2ABCG2
SCHEMBL7182545 0.87 ESR1 (0.52) ESR1ESR2ABCG2
SCHEMBL7190635 0.86 ESR1 (0.52) ESR1ESR2
SCHEMBL7190627 0.86 ESR1 (0.52) ESR1ESR2
SCHEMBL7182549 0.85 ESR1 (0.60) ESR1ESR2
SCHEMBL7182543 0.85 ESR1 (0.60) ESR1ESR2
SCHEMBL7183993 0.85 ESR1 (0.59) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP claimed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US claimed
EP-0835867-A1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-15 EP claimed
EP-0835867-B1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods LILLY CO ELI (US) 2003-12-03 EP disclosed
US-5916916-A USEFUL AS SELECTIVE ESTROGEN RECEPTOR MODULATORS. ELI LILLY AND COMPANY (US) 1999-06-29 US disclosed
EP-0835867-A1 1-Aryloxy-2-arylnaphthyl compounds, intermediates, compositions, and methods ELI LILLY AND COMPANY (US) 1998-04-15 EP disclosed