SCHEMBL7185986

SCHEMBL7185986

O=C(N[C@@H](CS(=O)(=O)c1ccc(Sc2ccccc2)cc1)C(=O)O)OCc1ccccc1

nearest known ligand 0.82

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 8/20 0.82
CA2 P00918 1/20 0.49
PPARA Q07869 3/20 0.47
CASP1 P29466 2/20 0.47
PPARG P37231 1/20 0.47
CTRB1 P17538 2/20 0.45
CTSL P07711 2/20 0.45
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
F2 P00734 1/20 0.45
PRSS1 P07477 1/20 0.45
PRSS2 P07478 1/20 0.45
PRSS3 P35030 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185980 1.00 MMP13 (0.82) MMP13CA2PPARACASP1PPARG
SCHEMBL7185942 0.90 MMP13 (0.67) MMP13CA2CASP1
SCHEMBL7185940 0.90 MMP13 (0.67) MMP13CA2CASP1
SCHEMBL7180333 0.85 MMP13 (0.82) MMP13CASP1CTSSCTSK
SCHEMBL7183683 0.82 MMP13 (0.79) MMP13
SCHEMBL7183687 0.82 MMP13 (0.79) MMP13
SCHEMBL22783671 0.79 PPARA (0.53) MMP13CA2PPARACASP1PPARG
SCHEMBL2749553 0.78 PPARA (0.53) MMP13CA2PPARACASP1PPARG
SCHEMBL7349434 0.78 CA12 (0.57) MMP13CA2PPARACASP1PPARG
SCHEMBL9686663 0.78 CA12 (0.57) MMP13CA2PPARACASP1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6583299-B1 Matrix metalloprotease inhibitors; nonsuppression of tumor necrosis factor production G.D. SEARLE & CO. 2003-06-24 US disclosed
EP-1178959-A1 ALPHA-AMINO-BETA-SULFONYL HYDROXAMIC ACID COMPOUNDS G.D. SEARLE & CO. (US) 2002-02-13 EP disclosed
WO-2000071514-A1 α-AMINO-β-SULFONYL HYDROXAMIC ACID COMPOUNDS G.D. SEARLE & CO. (US) 2000-11-30 WO disclosed