SCHEMBL7185940

SCHEMBL7185940

O=C(CNC(=O)OCc1ccccc1)NC(CS(=O)(=O)c1ccc(Sc2ccccc2)cc1)C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 9/20 0.67
MMP2 P08253 3/20 0.45
MMP9 P14780 3/20 0.45
CASP1 P29466 1/20 0.43
MAPK1 P28482 1/20 0.43
CA2 P00918 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MMP1 P03956 1/20 0.42
MMP3 P08254 1/20 0.42
MMP7 P09237 1/20 0.42
CYP3A4 P08684 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7185942 1.00 MMP13 (0.67) MMP13MMP2MMP9CASP1MAPK1
SCHEMBL7185980 0.90 MMP13 (0.82) MMP13CASP1CA2
SCHEMBL7185986 0.90 MMP13 (0.82) MMP13CASP1CA2
SCHEMBL31488862 0.77 ALDH1A1 (0.51) CASP1MAPK1ALDH1A1CYP3A4
SCHEMBL7183687 0.77 MMP13 (0.79) MMP13MMP2ALDH1A1MMP1MMP3
SCHEMBL8976911 0.77 CTSL (0.55) ALDH1A1
SCHEMBL7183683 0.77 MMP13 (0.79) MMP13MMP2ALDH1A1MMP1MMP3
SCHEMBL330061 0.77 CTSL (0.55) ALDH1A1
SCHEMBL31265234 0.77 CASP1 (0.54) CASP1MAPK1ALDH1A1
SCHEMBL5486969 0.77 CTSL (0.55) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6583299-B1 Matrix metalloprotease inhibitors; nonsuppression of tumor necrosis factor production G.D. SEARLE & CO. 2003-06-24 US disclosed