SCHEMBL7186449

SCHEMBL7186449

C=C1CC[C@H]2[C@@H]3CCc4c[c]ccc4[C@H]3CC[C@]12CC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 4/20 0.43
STS P08842 5/20 0.39
ESR1 P03372 7/20 0.37
ESR2 Q92731 5/20 0.37
LMNA P02545 4/20 0.37
HSD17B10 Q99714 4/20 0.37
SHBG P04278 3/20 0.37
MAPT P10636 3/20 0.37
AKR1B10 O60218 2/20 0.37
CYP1A2 P05177 2/20 0.37
PGR P06401 2/20 0.37
SERPINA6 P08185 2/20 0.37
CYP3A4 P08684 2/20 0.37
AR P10275 2/20 0.37
AKR1B1 P15121 2/20 0.37
SLC6A4 P31645 2/20 0.37
SNCA P37840 2/20 0.37
HTR2B P41595 2/20 0.37
BLM P54132 2/20 0.37
PMP22 Q01453 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7179669 0.87 HSD17B1 (0.58) HSD17B1STSESR1ESR2LMNA
SCHEMBL7175364 0.87 HSD17B1 (0.58) HSD17B1STSESR1ESR2LMNA
SCHEMBL7188971 0.86 HSD17B1 (0.42) HSD17B1STSESR1ESR2LMNA
SCHEMBL7188895 0.85 HSD17B1 (0.44) HSD17B1STSESR1ESR2LMNA
SCHEMBL8710195 0.83 STS (0.47) HSD17B1STSESR1ESR2LMNA
SCHEMBL7175660 0.81 HSD17B1 (0.48) HSD17B1STSESR1ESR2LMNA
SCHEMBL7175664 0.81 HSD17B1 (0.48) HSD17B1STSESR1ESR2LMNA
SCHEMBL7182171 0.79 HSD17B1 (0.42) HSD17B1STSESR1ESR2LMNA
SCHEMBL7187506 0.79 HSD17B1 (0.42) HSD17B1STSESR1ESR2LMNA
SCHEMBL6266816 0.78 SHBG (0.43) HSD17B1STSESR1ESR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6583130-B1 Substituted with acyl, oxycarbonyl, aminocarbonyl, sulfonyl, or aminosulfonyl; inhibit steroid sulfatase, do not exhibit any estrogenic effect and will not yield any estrogenic products on hydrolysis; treatment of estrogen-dependent tumors SCHERING AG (DE) 2003-06-24 US claimed
US-6583130-B1 Substituted with acyl, oxycarbonyl, aminocarbonyl, sulfonyl, or aminosulfonyl; inhibit steroid sulfatase, do not exhibit any estrogenic effect and will not yield any estrogenic products on hydrolysis; treatment of estrogen-dependent tumors SCHERING AG (DE) 2003-06-24 US disclosed