SCHEMBL7187232

SCHEMBL7187232

CS(=O)(=O)C(CCNC(=O)C(CNC(=O)N1CCOCC1)S(=O)(=O)Cc1ccccc1)C(=O)c1nc2ccccc2o1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.38
LIPC P11150 2/20 0.37
LIPG Q9Y5X9 2/20 0.37
KDM4E B2RXH2 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
HTT P42858 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
USP2 O75604 1/20 0.34
MAPK1 P28482 1/20 0.34
BRCA1 P38398 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7045925 0.90 CTSS (0.36) CTSSKDM4ECYP3A4CYP2C9HTT
SCHEMBL7045927 0.90 CTSS (0.38) CTSSLIPCLIPGKDM4ECYP3A4
SCHEMBL7114802 0.89 LMNA (0.38) CTSSKDM4EMEN1KMT2AALDH1A1
SCHEMBL6464598 0.87 CTSS (0.35) CTSSKDM4ECYP3A4CYP2C9HTT
SCHEMBL6464428 0.87 CTSS (0.39) CTSSCYP3A4CYP2C9
SCHEMBL7043175 0.85 DAGLA (0.46) CTSSLIPCLIPGKDM4EHTT
SCHEMBL7046398 0.85 XDH (0.38) CTSSKDM4ECYP3A4CYP2C9
SCHEMBL6467366 0.84 DAGLA (0.47) LIPCLIPGKDM4EHTTMEN1
SCHEMBL6463188 0.84 DAGLA (0.48) LIPCLIPGKDM4EHTTMEN1
SCHEMBL7044329 0.82 KDM4E (0.38) CTSSLIPCLIPGKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6576630-B1 Alkanoyl substituted benzooxazoles or naphthooxazoles AXYS PHARMACEUTICALS, INC. 2003-06-10 US disclosed