SCHEMBL7187629

SCHEMBL7187629

Cc1ccc(S(=O)(=O)N2CCC[C@H]2C(=O)N[C@@H](Cc2ccc(NS(=O)(=O)CCl)cc2)C(=O)O)cc1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.62
ITGA5 P08648 3/20 0.62
ITGA4 P13612 7/20 0.61
ITGAV P06756 3/20 0.56
ALDH1A1 P00352 1/20 0.54
MAPK1 P28482 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
ITGB7 P26010 1/20 0.51
FKBP1A P62942 1/20 0.50
ITGA2 P17301 1/20 0.50
TSHR P16473 1/20 0.49
PLAU P00749 1/20 0.49
HPN P05981 1/20 0.49
GAA P10253 1/20 0.48
HPGD P15428 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7325429 0.91 ITGA4 (0.56) ITGB1ITGA5ITGA4ITGAVMAPK1
SCHEMBL6709406 0.91 ITGB1 (0.64) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL5690742 0.89 ITGB1 (0.71) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL6712427 0.88 ITGA4 (0.65) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL7327937 0.88 ITGB1 (0.61) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL7322859 0.88 ITGB1 (0.61) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL6709558 0.88 ITGB1 (0.69) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL6708116 0.87 ITGB1 (0.60) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL6714530 0.87 ITGA4 (0.66) ITGB1ITGA5ITGA4ITGAVALDH1A1
SCHEMBL7069740 0.87 ALDH1A1 (0.70) ITGB1ITGA5ITGA4ITGAVALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6583139-B1 Treatment of inflammatory diseases; inflammatory brain diseases such as multiple sclerosis; N-(Toluene-4-sulfonyl)-L-prolyl-4-(alpha -methylbenzyloxy)-L-phenylalanine; Very Late Antigen 4 BIOGEN IDEC INTERNATIONAL HOLDING LTD. (BM) 2003-06-24 US claimed
US-6583139-B1 Treatment of inflammatory diseases; inflammatory brain diseases such as multiple sclerosis; N-(Toluene-4-sulfonyl)-L-prolyl-4-(alpha -methylbenzyloxy)-L-phenylalanine; Very Late Antigen 4 BIOGEN IDEC INTERNATIONAL HOLDING LTD. (BM) 2003-06-24 US disclosed