SCHEMBL71948

SCHEMBL71948

CCOC(=O)Cc1ccc(NC(=O)c2cn(C)c3ccccc23)c(C)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.48
MEN1 O00255 1/20 0.48
NPC1 O15118 1/20 0.48
KMT2A Q03164 1/20 0.48
MAPT P10636 3/20 0.48
POLB P06746 2/20 0.48
ITGB1 P05556 1/20 0.45
ITGA4 P13612 1/20 0.45
MAOB P27338 1/20 0.45
LMNA P02545 3/20 0.45
NR4A2 P43354 1/20 0.44
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CREBBP Q92793 1/20 0.43
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
TP53 P04637 1/20 0.41
CNR2 P34972 1/20 0.41
PTPN5 P54829 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2429129 0.90 ITGB1 (0.55) RAB9AKMT2AMAPTPOLBITGB1
SCHEMBL72718 0.89 MAPT (0.57) RAB9AMEN1KMT2AMAPTPOLB
SCHEMBL14505040 0.88 MAPT (0.45) RAB9AMEN1NPC1KMT2AMAPT
SCHEMBL70951 0.87 RAB9A (0.52) RAB9AMEN1NPC1KMT2AMAPT
SCHEMBL14591763 0.84 RAB9A (0.49) RAB9AMEN1NPC1KMT2AMAPT
SCHEMBL91593 0.83 RAB9A (0.52) RAB9AMEN1NPC1KMT2AMAPT
SCHEMBL92383 0.81 RAB9A (0.60) RAB9AMEN1NPC1KMT2AMAPT
SCHEMBL2432469 0.80 ALDH1A1 (0.44) RAB9AMEN1NPC1KMT2AMAPT
SCHEMBL3579447 0.80 ITGB1 (0.56) RAB9AMEN1NPC1KMT2AMAPT
SCHEMBL72352 0.76 POLB (0.61) MEN1KMT2AMAPTPOLBITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961750-B1 VLA-4 INHIBITORY DRUG DAIICHI SANKYO CO LTD (JP) 2013-09-18 EP disclosed