SCHEMBL7199134

SCHEMBL7199134

O=C(C#Cc1cccs1)c1ccccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 2/20 0.50
WNT3A P56704 2/20 0.50
RAB9A P51151 3/20 0.47
HPGD P15428 2/20 0.44
NPC1 O15118 3/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 3/20 0.41
ALOX15 P16050 1/20 0.41
PTPN1 P18031 1/20 0.38
ERCC5 P28715 1/20 0.38
FEN1 P39748 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 2/20 0.38
FFAR1 O14842 1/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29693871 1.00 CTNNB1 (0.50) CTNNB1WNT3ARAB9AHPGDNPC1
SCHEMBL7204989 0.84 CES2 (0.45) CTNNB1WNT3ARAB9AHPGDNPC1
SCHEMBL7199658 0.83 CES2 (0.41) CTNNB1WNT3ARAB9AHPGDNPC1
SCHEMBL7203229 0.81 TP53 (0.47) HPGDCES2CES1KDM4EALDH1A1
SCHEMBL7205541 0.81 CTNNB1 (0.56) CTNNB1WNT3ARAB9ANPC1ALDH1A1
SCHEMBL28672048 0.78 MAPK1 (0.43) RAB9AHPGDNPC1ALDH1A1MEN1
SCHEMBL7200524 0.77 ALDH1A1 (0.37) CTNNB1WNT3ARAB9AHPGDNPC1
SCHEMBL7202747 0.77 HSP90AA1 (0.49) RAB9AHPGDNPC1CES1KDM4E
SCHEMBL28745771 0.77 NPC1 (0.51) RAB9AHPGDNPC1KDM4EALDH1A1
SCHEMBL29625158 0.77 NPC1 (0.51) RAB9AHPGDNPC1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110256411-B Preparation method of 2, 3-disubstituted benzo-gamma-pyrone derivative 华侨大学 2022-06-07 CN disclosed
US-6605730-B2 3-(2-Thienyl)-5-phenyl-1H-pyrazole compounds of given formula NIHON BAYER AGROCHEM K.K. (JP) 2003-08-12 US disclosed
US-20030028034-A1 Nematicidal pyrazoles WADA KATSUAKI (JP) 2003-02-06 US disclosed
US-6310049-B1 3-(2-THIENYL),5-(SUBSTITUTED PHENYL)-1H-PYRAZOLES AND 3-(SUBSTITUTED PHENYL),5-(2-THIENYL)-1H-PYRAZOLES OF GIVEN FORMULA; ANTHELMINTICS NIHON BAYER AGROCHEM K.K. (JP) 2001-10-30 US disclosed
EP-1104418-A2 NEMATICIDAL PYRAZOLES NIHON BAYER AGROCHEM K.K. (JP) 2001-06-06 EP disclosed
WO-2000009500-A2 NEMATICIDAL PYRAZOLES NIHON BAYER AGROCHEM K.K. (JP) 2000-02-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030028034-A1 Nematicidal pyrazoles CBR3, CBR1, CCR4 CTNNB1 2248/4885WNT3A 2751/4885RAB9A 1643/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.