SCHEMBL7200439

SCHEMBL7200439

CC(=O)c1ccc(N2CCN(Cc3nc4c(C(N)=O)cccc4[nH]3)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AURKA O14965 2/20 0.57
AURKB Q96GD4 2/20 0.57
PARP1 P09874 13/20 0.51
NPC1 O15118 1/20 0.48
GAA P10253 1/20 0.48
KDR P35968 1/20 0.48
DRD4 P21917 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3582276 0.76 AURKB (0.82) AURKAAURKBPARP1KDR
SCHEMBL3580117 0.75 AURKB (0.77) AURKAAURKBPARP1KDR
SCHEMBL6841873 0.74 PARP1 (0.62) PARP1
SCHEMBL6964340 0.73 PARP1 (0.53) PARP1
SCHEMBL7479562 0.73 PARP1 (0.56) AURKBPARP1KDR
SCHEMBL3582843 0.73 AURKB (0.76) AURKAAURKBPARP1KDR
SCHEMBL3574435 0.73 AURKB (1.00) AURKAAURKBPARP1KDR
SCHEMBL3585484 0.72 PARP1 (0.75) AURKAAURKBPARP1KDR
SCHEMBL19002890 0.72 DRD4 (0.77) PARP1GAADRD4
SCHEMBL5620757 0.72 AURKA (0.67) AURKAAURKBPARP1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003106430-A1 BENZIMIDAZOLE INHIBITORS OF POLY(ADP-RIBOSYL) POLYMERASE PFIZER INC. (US) 2003-12-24 WO disclosed