SCHEMBL7201032

SCHEMBL7201032

O=C1c2ccccc2C(=O)N1C1CCC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.57
L3MBTL1 Q9Y468 1/20 0.51
TSHR P16473 3/20 0.49
CHRM2 P08172 1/20 0.49
OPRM1 P35372 1/20 0.49
DDB1 Q16531 1/20 0.49
CRBN Q96SW2 1/20 0.49
IKZF3 Q9UKT9 1/20 0.49
CYP1A2 P05177 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
KMT2A Q03164 1/20 0.48
HPGD P15428 2/20 0.47
HSD17B10 Q99714 2/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47
MC4R P32245 1/20 0.47
HTR2B P41595 2/20 0.46
TMEM97 Q5BJF2 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30212234 1.00 ALDH1A1 (0.57) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
SCHEMBL18935574 0.96 ALDH1A1 (0.62) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
SCHEMBL23967443 0.94 ALDH1A1 (0.65) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
SCHEMBL30987468 0.94 ALDH1A1 (0.65) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
SCHEMBL2653818 0.94 ALDH1A1 (0.65) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
SCHEMBL2665681 0.91 L3MBTL1 (0.54) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
SCHEMBL9625796 0.91 L3MBTL1 (0.54) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
Bicarbonate SCHEMBL14811674 0.87 ALDH1A1 (0.58) ALDH1A1L3MBTL1TSHRTDP1KMT2A
SCHEMBL8477142 0.85 ALDH1A1 (0.49) ALDH1A1L3MBTL1TSHRCHRM2OPRM1
SCHEMBL14075773 0.84 ALDH1A1 (0.50) ALDH1A1L3MBTL1TDP1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109180558-A It is the method that one step of starting material constructs N- cyclobutyl phthalimide using imines 桂林理工大学 2019-01-11 CN claimed
US-11673900-B2 Process for preparing 7H-pyrrolo[2,3-d]pyrimidine derivatives and synthetic intermediates thereof JAPAN TOBACCO INC. (JP) 2023-06-13 US disclosed
US-20200216470-A1 PROCESS FOR PREPARING 7H-PYRROLO[2,3-d]PYRIMIDINE DERIVATIVES AND SYNTHETIC INTERMEDIATES THEREOF JAPAN TOBACCO INC. (JP) 2020-07-09 US disclosed
CN-109180558-A It is the method that one step of starting material constructs N- cyclobutyl phthalimide using imines 桂林理工大学 2019-01-11 CN disclosed
CN-109180558-A It is the method that one step of starting material constructs N- cyclobutyl phthalimide using imines 桂林理工大学 2019-01-11 CN disclosed
CN-109180558-A It is the method that one step of starting material constructs N- cyclobutyl phthalimide using imines 桂林理工大学 2019-01-11 CN disclosed
WO-2017040606-A1 ISOXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PULMONARY DISEASES AND DISORDERS PROTEOSTASIS THERAPEUTICS, INC. (US) 2017-03-09 WO disclosed
EP-1071645-A4 PHOSPHODIESTERASE ISOENZYME DENOMINATED 4 (PDE 4) INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2003-04-02 EP disclosed
EP-1071645-A1 PHOSPHODIESTERASE ISOENZYME DENOMINATED 4 (PDE 4) INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-31 EP disclosed
US-6172118-B1 Compounds SMITHKLINE BEECHAM CORPORATION 2001-01-09 US disclosed
WO-1999052847-A1 PHOSPHODIESTERASE ISOENZYME DENOMINATED 4 (PDE 4) INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11673900-B2 Process for preparing 7H-pyrrolo[2,3-d]pyrimidine derivatives and synthetic intermediates thereof JAK1, JAK3, JAK2 ALDH1A1 1674/4885L3MBTL1 3776/4885TSHR 2651/4885
US-20200216470-A1 PROCESS FOR PREPARING 7H-PYRROLO[2,3-d]PYRIMIDINE DERIVATIVES AND SYNTHETIC INTERMEDIATES THEREOF JAK1, JAK3, JAK2 ALDH1A1 1674/4885L3MBTL1 3776/4885TSHR 2651/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.