SCHEMBL7201362

SCHEMBL7201362

Cc1cc(N(C(=O)[C@@H]2CCCN2C(=O)[C@@H](NC(=O)[C@H](CC(=O)O)NC(=O)[C@H](CC(C)C)NC(=O)Cc2ccccc2)C(C)C)[C@@H](CO)C(=O)O)ccc1NC(N)=O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 7/20 0.43
ITGA4 P13612 7/20 0.43
CALCRL Q16602 3/20 0.41
CTSD P07339 7/20 0.40
CTSE P14091 7/20 0.40
BACE1 P56817 4/20 0.40
EPHA2 P29317 2/20 0.39
AKT1 P31749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7195991 0.87 CALCRL (0.46) ITGB1ITGA4CALCRLCTSDCTSE
SCHEMBL8334047 0.81 CALCRL (0.49) ITGB1ITGA4CALCRLCTSDCTSE
SCHEMBL5208748 0.80 CTSD (0.49) ITGB1ITGA4CALCRLCTSDCTSE
SCHEMBL1223367 0.77 ITGB1 (0.64) ITGB1ITGA4
SCHEMBL13035172 0.76 ITGB1 (0.63) ITGB1ITGA4
SCHEMBL7202828 0.76 ITGB1 (0.41) ITGB1ITGA4
SCHEMBL7197725 0.74 ITGB1 (0.41) ITGB1ITGA4CTSDBACE1
SCHEMBL7197381 0.74 ITGB1 (0.41) ITGB1ITGA4CTSDBACE1
SCHEMBL2045662 0.73 REN (0.54) CTSDCTSEBACE1
SCHEMBL7419554 0.73 REN (0.54) CTSDCTSEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596687-B1 For treatment of many inflammatory and autoimmune diseases BIOGEN, INC. 2003-07-22 US claimed