SCHEMBL7202389

SCHEMBL7202389

COc1ccccc1-c1c(C#N)c(N)nc2cc(-c3ccc(CN4CCS(O)(O)CC4)cc3)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 5/20 0.43
HPGD P15428 5/20 0.43
HSD17B10 Q99714 3/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
BLM P54132 1/20 0.42
LMNA P02545 3/20 0.41
MAPT P10636 2/20 0.41
ATM Q13315 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
SRC P12931 6/20 0.41
FYN P06241 2/20 0.41
DHFR P00374 1/20 0.40
TSHR P16473 2/20 0.39
EGFR P00533 1/20 0.39
MAP2K1 Q02750 1/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MAPK1 P28482 1/20 0.39
S1PR4 O95977 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7202383 0.79 JAK1 (0.47) ALDH1A1HPGDHSD17B10MEN1KMT2A
SCHEMBL7166273 0.78 SRC (0.53) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7202387 0.75 JAK1 (0.44) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL7149809 0.72 ALDH1A1 (0.43) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL6223729 0.72 ALDH1A1 (0.67) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL16618012 0.70 RIOK3 (0.54) ALDH1A1KDM4EHPGDSRCFYN
SCHEMBL7913439 0.68 KDM4E (0.60) ALDH1A1KDM4EHPGDHSD17B10MEN1
SCHEMBL3220989 0.68 SRC (0.84) SRCFYNEGFRMAP2K1
SCHEMBL7166266 0.66 SRC (0.52) SRCFYNEGFRMAP2K1
SCHEMBL27576302 0.64 KDM4E (0.49) ALDH1A1KDM4EHPGDHSD17B10MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268431-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS Wyeth (US) 2003-01-02 EP disclosed
WO-2001072711-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH (US) 2001-10-04 WO disclosed