SCHEMBL7149809

SCHEMBL7149809

CCN1CCN(c2ccc(-c3ccc4c(-c5ccccc5OC)c(C#N)c(N)nc4c3)nc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
KDM4E B2RXH2 5/20 0.43
HSD17B10 Q99714 2/20 0.43
HPGD P15428 4/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
BLM P54132 1/20 0.41
MAPT P10636 3/20 0.40
LMNA P02545 2/20 0.40
ATM Q13315 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
TSHR P16473 1/20 0.40
DHFR P00374 1/20 0.38
PKM P14618 1/20 0.38
MAPK1 P28482 1/20 0.38
PRKDC P78527 1/20 0.38
PDE3A Q14432 1/20 0.38
S1PR4 O95977 1/20 0.37
GLA P06280 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7149801 0.88 PIP4K2A (0.44) ALDH1A1KDM4EHSD17B10HPGDMEN1
SCHEMBL7149804 0.83 LMNA (0.39) ALDH1A1KDM4EHSD17B10HPGDMEN1
SCHEMBL7166273 0.75 SRC (0.53) ALDH1A1KDM4EHSD17B10HPGDMEN1
SCHEMBL7202389 0.72 ALDH1A1 (0.43) ALDH1A1KDM4EHSD17B10HPGDMEN1
SCHEMBL6223729 0.70 ALDH1A1 (0.67) ALDH1A1KDM4EHSD17B10HPGDMEN1
SCHEMBL16618012 0.70 RIOK3 (0.54) ALDH1A1KDM4EHPGDCHEK1SRC
SCHEMBL3224685 0.70 SRC (0.74) SRC
SCHEMBL28750720 0.67 ADORA2A (0.51) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL7913439 0.66 KDM4E (0.60) ALDH1A1KDM4EHSD17B10HPGDMEN1
SCHEMBL27576302 0.65 KDM4E (0.49) ALDH1A1KDM4EHSD17B10HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268431-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS Wyeth (US) 2003-01-02 EP disclosed
WO-2001072711-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH (US) 2001-10-04 WO disclosed