SCHEMBL7166273

SCHEMBL7166273

COc1ccccc1-c1c(C#N)c(N)nc2cc(-c3cc(CN4CCOCC4)ccn3)ccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 10/20 0.53
EGFR P00533 2/20 0.42
FYN P06241 1/20 0.42
MAP2K1 Q02750 1/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
MEN1 O00255 1/20 0.40
BLM P54132 1/20 0.40
KMT2A Q03164 1/20 0.40
LRRK2 Q5S007 1/20 0.40
CDK1 P06493 1/20 0.40
CDK2 P24941 1/20 0.40
CASP3 P42574 1/20 0.40
CDK9 P50750 1/20 0.40
CASP7 P55210 1/20 0.40
PDE4B Q07343 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7166266 0.88 SRC (0.52) SRCEGFRFYNMAP2K1JAK2
SCHEMBL7166270 0.83 SRC (0.48) SRCEGFRFYNMAP2K1JAK2
SCHEMBL7202389 0.78 ALDH1A1 (0.43) SRCEGFRFYNMAP2K1KDM4E
SCHEMBL7149809 0.75 ALDH1A1 (0.43) SRCKDM4EALDH1A1HPGDHSD17B10
SCHEMBL6223729 0.70 ALDH1A1 (0.67) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL3232975 0.70 SRC (1.00) SRCEGFRFYNMAP2K1
SCHEMBL16618012 0.68 RIOK3 (0.54) SRCEGFRFYNMAP2K1KDM4E
SCHEMBL28748064 0.67 SRC (0.62) SRCEGFRFYNMAP2K1JAK2
SCHEMBL7692261 0.66 ADORA2A (0.45) KDM4EALDH1A1HPGDHSD17B10MEN1
SCHEMBL4765678 0.66 DRD2 (0.53) ALDH1A1JAK2JAK1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268431-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS Wyeth (US) 2003-01-02 EP disclosed
WO-2001072711-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH (US) 2001-10-04 WO disclosed