SCHEMBL7202439

SCHEMBL7202439

CN1CC=C(c2cc3ccccc3[nH]2)CC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.51
SLC6A4 P31645 2/20 0.51
KDM4E B2RXH2 1/20 0.51
LMNA P02545 1/20 0.51
POLB P06746 1/20 0.51
HTR1A P08908 1/20 0.51
ALOX15 P16050 1/20 0.51
HSD17B10 Q99714 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
HRH4 Q9H3N8 1/20 0.43
QDPR P09417 2/20 0.43
KDR P35968 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7859752 0.82 SLC6A4 (0.56) HTR6SLC6A4HRH4
Bromide SCHEMBL7868021 0.81 SLC6A4 (0.52) HTR6SLC6A4QDPR
SCHEMBL7496144 0.81 HRH4 (0.46) HTR6SLC6A4HRH4QDPR
SCHEMBL6646297 0.81 TNKS (0.51) HTR6SLC6A4KDM4ELMNAPOLB
SCHEMBL11864700 0.80 QDPR (0.49) LMNAHRH4QDPRKDR
SCHEMBL7866268 0.79 SLC6A4 (0.44) HTR6SLC6A4KDM4ELMNAPOLB
Bromide SCHEMBL7867418 0.77 HRH4 (0.45) SLC6A4HRH4
SCHEMBL7866398 0.77 DRD2 (0.61) HTR6HTR1AKDR
Bromide SCHEMBL7859817 0.77 HTR6 (0.50) HTR6SLC6A4KDM4ELMNAPOLB
SCHEMBL7214674 0.74 DRD2 (0.42) SLC6A4HTR1AHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6608079-B1 Activating serotonin-1F receptors, inhibiting neuronal protein extravasation, treating migraine ELI LILLY AND COMPANY 2003-08-19 US disclosed
EP-1196380-A2 INDOLES AND INDAZOLES FOR THE TREATMENT OF MIGRAINE NPS Allelix Corp. (CA) 2002-04-17 EP disclosed
WO-2001005758-A2 INDOLES AND INDAZOLES FOR THE TREATMENT OF MIGRAINE NPS ALLELIX CORP. (CA) 2001-01-25 WO disclosed