Ly-293284

Ly-293284

SCHEMBL7202815

CCCN(CCC)C1Cc2c[nH]c3ccc(C(C)=O)c(c23)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 1.00
HTR1D P28221 5/20 0.65
HTR1B P28222 5/20 0.65
DRD2 P14416 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ly-293284 SCHEMBL6902000 1.00 HTR1A (1.00) HTR1AHTR1DHTR1BDRD2
Ly-293284 SCHEMBL7204055 1.00 HTR1A (1.00) HTR1AHTR1DHTR1BDRD2
SCHEMBL9412130 0.91 HTR1A (0.83) HTR1AHTR1DHTR1BDRD2
SCHEMBL8889776 0.91 HTR1A (0.83) HTR1AHTR1DHTR1BDRD2
SCHEMBL6364891 0.90 HTR1A (0.81) HTR1AHTR1DHTR1BDRD2
SCHEMBL6765275 0.90 HTR1A (0.81) HTR1AHTR1DHTR1BDRD2
SCHEMBL7208944 0.90 HTR1A (0.81) HTR1AHTR1DHTR1BDRD2
SCHEMBL8983347 0.90 HTR1A (0.81) HTR1AHTR1DHTR1BDRD2
Acetic Acid SCHEMBL7513634 0.89 HTR1A (0.80) HTR1AHTR1DHTR1BDRD2
SCHEMBL7516908 0.89 HTR1A (0.80) HTR1AHTR1DHTR1BDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023212244-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS, INC. (US) 2023-11-02 WO claimed
EP-3953000-A1 CELL MEMBRANE PERMEABILITY RESTORING THERAPY Shine, Ian Basil (US) 2022-02-16 EP claimed
EP-0471576-B1 6-substituted-tetrahydrobenz[cd]indoles LILLY CO ELI (US) 2003-03-12 EP claimed
US-5292766-A Method for improving primary memory and/or learning ELI LILLY AND COMPANY (US) 1994-03-08 US claimed
EP-0565274-A1 5-Ht1A agonists for improving primary memory and/or learning ELI LILLY AND COMPANY (US) 1993-10-13 EP claimed
US-5229409-A Antidepressant, tranquilizer ELI LILLY AND COMPANY (US) 1993-07-20 US claimed
JP-4230663-A None JP disclosed
WO-2023212244-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS, INC. (US) 2023-11-02 WO disclosed
EP-0471576-B1 6-substituted-tetrahydrobenz[cd]indoles LILLY CO ELI (US) 2003-03-12 EP disclosed
US-5292766-A Method for improving primary memory and/or learning ELI LILLY AND COMPANY (US) 1994-03-08 US disclosed
EP-0565274-A1 5-Ht1A agonists for improving primary memory and/or learning ELI LILLY AND COMPANY (US) 1993-10-13 EP disclosed
US-5229409-A Antidepressant, tranquilizer ELI LILLY AND COMPANY (US) 1993-07-20 US disclosed
JP-H04230663-A 6-SUBSTITUTED TETRAHYDROBENZ(C,D)INDOLE ELI LILLY & CO 1992-08-19 JP disclosed