SCHEMBL7202899

SCHEMBL7202899

COc1ccc(C(Nc2ncnc3c2ncn3[C@H]2C[C@@H](OC(=O)c3ccccc3)[C@H](C(O)C(c3ccccc3)(c3ccccc3)c3ccc(OC)cc3)O2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.41
ADORA2B P29275 2/20 0.41
ADORA3 P0DMS8 2/20 0.38
ADORA1 P30542 1/20 0.37
PRKAG1 P54619 1/20 0.37
PRKAA1 Q13131 1/20 0.37
PRKAB1 Q9Y478 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532594 0.86 POLB (0.41) ADORA2AADORA2BADORA1
SCHEMBL532593 0.85 TYMP (0.46) ADORA2AADORA2BADORA1
Hydroquinone SCHEMBL7070523 0.84 PRMT6 (0.41) ADORA2AADORA2BADORA3ADORA1PRKAG1
SCHEMBL4434106 0.84 ADORA2A (0.39) ADORA2AADORA2BADORA3ADORA1PRKAG1
SCHEMBL888001 0.83 ADORA3 (0.45) ADORA2AADORA2BADORA3ADORA1PRKAG1
SCHEMBL7075967 0.82 ADORA2B (0.39) ADORA2AADORA2BADORA3ADORA1
SCHEMBL7873202 0.82 ADORA2A (0.42) ADORA2AADORA2BADORA3ADORA1PRKAG1
SCHEMBL7879389 0.80 CHKA (0.36) ADORA2AADORA2BADORA3ADORA1
SCHEMBL2112347 0.78 ADORA3 (0.47) ADORA2AADORA2BADORA3ADORA1
SCHEMBL21577261 0.77 TYMP (0.46) ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6569837-B1 Administering 2'-deoxy-beta-L-erythro-pentofuranonucleoside alone or with another anti-hepatitis B agent such as 3TC (beta-L-2-hydroxymethyl-5-(cytosin-1-yl)-1,3-oxathiolane); use of beta-l-thymidine (telbivudine) IDENIX PHARMACEUTICALS INC. 2003-05-27 US disclosed