SCHEMBL7202949

SCHEMBL7202949

CC1(C)O[C@@H]2[C@H](O1)[C@@H](CO)O[C@H]2n1cnc2c(NCCc3ccccc3)nc(Cl)nc21

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 6/20 0.66
ADORA3 P0DMS8 6/20 0.66
ADORA2A P29274 5/20 0.66
PGK1 P00558 3/20 0.60
PGK2 P07205 3/20 0.60
NT5E P21589 2/20 0.58
TSHR P16473 2/20 0.57
NFKB1 P19838 1/20 0.57
THPO P40225 1/20 0.57
ADORA2B P29275 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7202938 1.00 ADORA1 (0.66) ADORA1ADORA3ADORA2APGK1PGK2
SCHEMBL5055239 0.95 ADORA1 (0.60) ADORA1ADORA3ADORA2APGK1PGK2
SCHEMBL19366689 0.91 ADORA3 (0.60) ADORA1ADORA3ADORA2ANT5EADORA2B
SCHEMBL25090698 0.91 ADORA3 (0.60) ADORA1ADORA3ADORA2ANT5EADORA2B
SCHEMBL5062524 0.89 ADORA3 (0.73) ADORA1ADORA3ADORA2APGK1PGK2
SCHEMBL7203455 0.85 PI4KA (0.53) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL7203458 0.85 PI4KA (0.53) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL31201331 0.85 ADORA1 (0.88) ADORA1ADORA3ADORA2APGK1PGK2
SCHEMBL24601292 0.84 ADORA3 (0.62) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL13238338 0.84 ADORA3 (0.73) ADORA1ADORA3ADORA2ATSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610665-B1 Treatment of inflammatory diseases, asthma or chronic obstructive pulmonary disease SMITHKLINE BEECHAM CORPORATION 2003-08-26 US disclosed
EP-1056759-B1 2-(PURIN-9-YL) -TETRAHYDROFURAN-3, 4-DIOL DERIVATIVES GLAXO GROUP LTD (GB) 2002-09-04 EP disclosed