SCHEMBL7203087

SCHEMBL7203087

C#CC(O)c1ccc(C(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 2/20 0.40
HTT P42858 2/20 0.40
PYCR1 P32322 1/20 0.40
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
CYP2C9 P11712 3/20 0.36
HIF1A Q16665 2/20 0.36
ALOX5 P09917 1/20 0.36
CYP2D6 P10635 1/20 0.36
TRPA1 O75762 1/20 0.35
PTGS1 P23219 1/20 0.35
CACNA1C Q13936 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPK1 P28482 1/20 0.35
UGT2B7 P16662 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
ALOX12 P18054 1/20 0.34
IDO1 P14902 1/20 0.34
USP5 P45974 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29184903 0.87 ESR1 (0.46) ESR1ESR2
SCHEMBL7199129 0.81 CHRNA7 (0.39) ESR1ESR2ALOX5ALDH1A1LMNA
SCHEMBL6957145 0.81 MAPT (0.38) HTTESR1ESR2HIF1AKDM4E
SCHEMBL1920526 0.81 TSHR (0.41) ESR1ESR2CYP2C9HIF1ACYP2D6
SCHEMBL6962580 0.78 ESR1 (0.62) TYRESR1ESR2CYP2C9HIF1A
SCHEMBL132554 0.76 AOC3 (0.38) HTTESR1ESR2ALOX5KDM4E
SCHEMBL12469442 0.76 AOC3 (0.38) HTTESR1ESR2ALOX5KDM4E
SCHEMBL3096700 0.76 PYCR1 (0.40) PYCR1ESR1ESR2ALOX5
SCHEMBL8019231 0.76 TSHR (0.60) TYRHTTESR1ESR2CYP2C9
SCHEMBL7199112 0.76 ESR1 (0.38) PYCR1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6605730-B2 3-(2-Thienyl)-5-phenyl-1H-pyrazole compounds of given formula NIHON BAYER AGROCHEM K.K. (JP) 2003-08-12 US disclosed
US-20030028034-A1 Nematicidal pyrazoles WADA KATSUAKI (JP) 2003-02-06 US disclosed
US-6310049-B1 3-(2-THIENYL),5-(SUBSTITUTED PHENYL)-1H-PYRAZOLES AND 3-(SUBSTITUTED PHENYL),5-(2-THIENYL)-1H-PYRAZOLES OF GIVEN FORMULA; ANTHELMINTICS NIHON BAYER AGROCHEM K.K. (JP) 2001-10-30 US disclosed
EP-1104418-A2 NEMATICIDAL PYRAZOLES NIHON BAYER AGROCHEM K.K. (JP) 2001-06-06 EP disclosed
WO-2000009500-A2 NEMATICIDAL PYRAZOLES NIHON BAYER AGROCHEM K.K. (JP) 2000-02-24 WO disclosed
EP-0360091-B1 PROCESS FOR THE PREPARATION OF ALKYL-SUBSTITUTED CINNAMIC ALDEHYDES BASF Aktiengesellschaft (DE) 1992-09-02 EP disclosed
US-4996365-A Preparation of alkyl-substituted cinnamaldehydes BASF AKTIENGESELLSCHAFT (DE) 1991-02-26 US disclosed
EP-0360091-A2 Process for the preparation of alkyl-substituted cinnamic aldehydes BASF Aktiengesellschaft (DE) 1990-03-28 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030028034-A1 Nematicidal pyrazoles CBR3, CBR1, CCR4 TYR 789/4885HTT 3125/4885PYCR1 248/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.