SCHEMBL7203845

SCHEMBL7203845

CC1(C)O[C@@H]2C(CO)OC(n3cnc4c(NCCC5CCCCC5)nc(Cl)nc43)[C@@H]2O1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.53
ADORA2B P29275 3/20 0.53
ADORA3 P0DMS8 3/20 0.53
ADORA1 P30542 3/20 0.53
MEN1 O00255 1/20 0.53
CYP1A2 P05177 1/20 0.53
MAPK1 P28482 1/20 0.53
KMT2A Q03164 1/20 0.53
RXFP1 Q9HBX9 1/20 0.52
PI4KA P42356 1/20 0.50
PI4K2B Q8TCG2 1/20 0.50
PI4K2A Q9BTU6 1/20 0.50
PI4KB Q9UBF8 1/20 0.50
ALOX15 P16050 1/20 0.50
HTR2C P28335 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7203847 1.00 ADORA2A (0.53) ADORA2AADORA2BADORA3ADORA1MEN1
SCHEMBL7203458 0.86 PI4KA (0.53) ADORA2AADORA2BADORA3ADORA1MEN1
SCHEMBL7203455 0.86 PI4KA (0.53) ADORA2AADORA2BADORA3ADORA1MEN1
SCHEMBL20180024 0.85 ADORA3 (0.72) ADORA2AADORA2BADORA3ADORA1MEN1
SCHEMBL8818648 0.83 ADORA1 (0.61) ADORA1PI4KAPI4K2BPI4K2API4KB
SCHEMBL7202938 0.82 ADORA1 (0.66) ADORA2AADORA2BADORA3ADORA1
SCHEMBL7202949 0.82 ADORA1 (0.66) ADORA2AADORA2BADORA3ADORA1
SCHEMBL25090698 0.80 ADORA3 (0.60) ADORA2AADORA2BADORA3ADORA1
SCHEMBL6574020 0.80 ADORA3 (0.66) ADORA2AADORA2BADORA3ADORA1MEN1
SCHEMBL19366689 0.80 ADORA3 (0.60) ADORA2AADORA2BADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610665-B1 Treatment of inflammatory diseases, asthma or chronic obstructive pulmonary disease SMITHKLINE BEECHAM CORPORATION 2003-08-26 US disclosed
EP-1056759-B1 2-(PURIN-9-YL) -TETRAHYDROFURAN-3, 4-DIOL DERIVATIVES GLAXO GROUP LTD (GB) 2002-09-04 EP disclosed