SCHEMBL7204913

SCHEMBL7204913

CC(C)C[C@H](N)C(=O)N(Cc1ccc(C#N)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36
MAOB P27338 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
NSD2 O96028 1/20 0.36
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
MMP2 P08253 1/20 0.34
ABCB1 P08183 3/20 0.34
ADAM17 P78536 1/20 0.34
EPHX2 P34913 1/20 0.33
TAS2R14 Q9NYV8 1/20 0.33
TRPA1 O75762 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1009189 0.83 NSD2 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4MAOB
SCHEMBL8771989 0.83 MMP2 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4MAOB
SCHEMBL6424007 0.81 NSD2 (0.43) MAOBNSD2CHRM2CHRM1CHRM3
SCHEMBL7465397 0.76 TSHR (0.44) CHRNB2CHRNB4CHRNA3CHRNA4MAOB
SCHEMBL2586342 0.76 SLC6A2 (0.44) MLYCDCHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL2578969 0.76 NSD2 (0.41) MLYCDCHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL7233237 0.74 NSD2 (0.53) SLC6A4NSD2CHRM2CHRM1CHRM3
SCHEMBL10712025 0.74 ANPEP (0.41)
SCHEMBL8773630 0.73 SLC7A5 (0.36)
SCHEMBL1737432 0.72 AKT1 (0.42) CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030153506-A1 Combination product comprising melagatran and factor VIIa inhibitor ASTRAZENECA AB (SE) 2003-08-14 US disclosed