Maleic Acid

Maleic Acid

SCHEMBL720767

C=C(C)C(=O)OCC.C=C(C)C(=O)OCC.O=C(O)/C=C\C(=O)O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 5/20 0.57
THRB P10828 1/20 0.52
TSHR P16473 4/20 0.46
GLO1 Q04760 1/20 0.45
ALDH1A1 P00352 7/20 0.44
LMNA P02545 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 1/20 0.41
CYP2D6 P10635 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL15653018 1.00 HCAR2 (0.57) HCAR2THRBTSHRGLO1ALDH1A1
Fumaric Acid SCHEMBL8953356 1.00 HCAR2 (0.57) HCAR2THRBTSHRGLO1ALDH1A1
Acrylic Acid SCHEMBL27651708 0.88 THRB (0.52) HCAR2THRBTSHRGLO1ALDH1A1
Acrylic Acid SCHEMBL265149 0.88 THRB (0.52) HCAR2THRBTSHRGLO1ALDH1A1
Acetic Acid SCHEMBL28298395 0.87 THRB (0.59) THRBTSHRGLO1ALDH1A1LMNA
Bicarbonate SCHEMBL10996730 0.87 THRB (0.59) THRBTSHRGLO1ALDH1A1LMNA
SCHEMBL15030 0.87
SCHEMBL19409375 0.87 THRB (0.64) THRBTSHRGLO1ALDH1A1LMNA
Acrylic Acid SCHEMBL23825514 0.86 THRB (0.50) HCAR2THRBTSHRGLO1ALDH1A1
Acrolein SCHEMBL11765226 0.85 HCAR2 (0.43) HCAR2THRBTSHRGLO1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 83 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210214573-A1 PHOTOPOLYMERIZABLE TYPE DENTAL SURFACE COATING COMPOSITION SHOFU INC. (JP) 2021-07-15 US disclosed
US-20200253835-A1 Dental Curable Composition TOKUYAMA DENTAL CORPORATION (JP) 2020-08-13 US disclosed
EP-3682862-A1 CURABLE DENTAL COMPOSITION Tokuyama Dental Corporation (JP) 2020-07-22 EP disclosed
EP-1704845-B1 Polymerization initiator composition for dental or surgical adhesive compositions SUN MEDICAL CO LTD (JP) 2019-07-03 EP disclosed
EP-2902007-B1 DENTAL FILLING REPAIRING MATERIAL TOKUYAMA DENTAL CORP (JP) 2019-01-09 EP disclosed
US-9192693-B2 Method for treatment of emphysema TERUMO KABUSHIKI KAISHA (JP) 2015-11-24 US disclosed
US-20150272833-A1 Dental Restorative Material TOKUYAMA DENTAL CORPORATION (JP) 2015-10-01 US disclosed
EP-2902007-A1 DENTAL FILLING REPAIRING MATERIAL Tokuyama Dental Corporation (JP) 2015-08-05 EP disclosed
EP-2809688-A1 LASER ENGRAVEABLE COMPOSITIONS FOR RELIEF IMAGE PRINTING ELEMENTS NAPP SYSTEMS, INC. (US) 2014-12-10 EP disclosed
WO-2013116011-A1 LASER ENGRAVEABLE COMPOSITIONS FOR RELIEF IMAGE PRINTING ELEMENTS NAPP SYSTEMS, INC. (US) 2013-08-08 WO disclosed
US-5021321-A Photothermography; antifogging agents; contrast; lamination of matrix of silver salts and reducing agent and dispersed particles of dye, polymer precursor and photoinitiator CANON KABUSHIKI KAISHA (JP) 1991-06-04 US disclosed
US-5001032-A Photosensitive material containing a photosensitive and heat developable element and a polymerizable layer and image-forming method utilizing the same CANON KABUSHIKI KAISHA (JP) 1991-03-19 US disclosed
EP-0412851-A2 Photosensitive member and multi-color image forming method CANON KABUSHIKI KAISHA (JP) 1991-02-13 EP disclosed
EP-0410803-A2 Image forming device CANON KABUSHIKI KAISHA (JP) 1991-01-30 EP disclosed
EP-0363790-A2 Image forming method and image forming medium CANON KABUSHIKI KAISHA (JP) 1990-04-18 EP disclosed
EP-0360014-A1 Photosensitive material and image forming method using same CANON KABUSHIKI KAISHA (JP) 1990-03-28 EP disclosed
EP-0332455-A2 Photosensitive material and image forming method CANON KABUSHIKI KAISHA (JP) 1989-09-13 EP disclosed
EP-0330504-A2 Photosensitive material and image forming method CANON KABUSHIKI KAISHA (JP) 1989-08-30 EP disclosed
EP-0328364-A2 Photosensitive material CANON KABUSHIKI KAISHA (JP) 1989-08-16 EP disclosed
EP-0326424-A2 Photosensitive composition, photosensitive material, and image forming method CANON KABUSHIKI KAISHA (JP) 1989-08-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200253835-A1 Dental Curable Composition SP1, H1-0, ERH HCAR2 993/4885THRB 1005/4885TSHR 2813/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.