SCHEMBL7207777

SCHEMBL7207777

Nc1ccc([N+](=O)[O-])cc1-c1nnn[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 7/20 0.45
MAPT P10636 5/20 0.45
CYP3A4 P08684 5/20 0.44
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
KDM4E B2RXH2 2/20 0.43
ALOX12 P18054 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
GAA P10253 1/20 0.42
THRB P10828 1/20 0.42
TSHR P16473 1/20 0.42
CAPN9 O14815 1/20 0.42
CASP3 P42574 1/20 0.42
PTPRC P08575 1/20 0.41
S100A4 P26447 1/20 0.41
MCL1 Q07820 1/20 0.41
HTT P42858 1/20 0.41
LMNA P02545 2/20 0.40
ALOX15 P16050 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2738746 0.88 CYP3A4 (0.47) TDP1MAPTCYP3A4ALDH1A1MEN1
SCHEMBL30389282 0.82 MAPT (0.58) TDP1MAPTCYP3A4ALDH1A1MEN1
SCHEMBL12821539 0.82 KDM4E (0.49) TDP1MAPTCYP3A4ALDH1A1MEN1
SCHEMBL31377032 0.82 KDM4E (0.49) TDP1MAPTCYP3A4ALDH1A1MEN1
SCHEMBL21051804 0.80 ALDH1A1 (0.49) TDP1MAPTCYP3A4ALDH1A1MEN1
SCHEMBL6775625 0.79 MAPT (0.50) TDP1MAPTALDH1A1MEN1KMT2A
SCHEMBL11684415 0.76 TDP1 (0.65) TDP1MAPTCYP3A4ALDH1A1MEN1
SCHEMBL264644 0.76 XDH (0.51) TDP1MAPTMEN1KMT2AGAA
SCHEMBL5311953 0.75 MAPT (0.60) TDP1MAPTCYP3A4ALDH1A1MEN1
SCHEMBL3277817 0.74 IDO1 (0.35) NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977741-B1 SUBSTITUTED PHENYL DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH AS (DK) 2003-09-03 EP disclosed
US-6297261-B1 POTENT CHLORIDE CHANNEL BLOCKERS; TREATMENT OF SICKLE CELL ANEMIA, BRAIN EDEMA FOLLOWING ISCHAEMIA OR TUMORS, DIARRHEA, HYPERTENSION (DIURETIC), OSTEOPOROSIS, AND FOR THE REDUCTION OF THE INTRAOCULAR PRESSURE NEUROSEARCH A/S (DK) 2001-10-02 US disclosed
US-4286090-A BLOWING AGENTS; PROPELLANTS; EXPLOSIVES; IGNITERS THE DOW CHEMICAL COMPANY (US) 1981-08-25 US disclosed