SCHEMBL7208466

SCHEMBL7208466

COc1ccc(S(=O)(=O)C2CCCC(S)C2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 4/20 1.00
MMP8 P22894 3/20 1.00
MMP1 P03956 2/20 1.00
ADAM17 P78536 3/20 0.68
MMP2 P08253 3/20 0.47
MMP9 P14780 3/20 0.47
PKM P14618 2/20 0.43
ELOVL6 Q9H5J4 1/20 0.41
HTT P42858 1/20 0.41
NPC1 O15118 1/20 0.41
PKLR P30613 1/20 0.41
RAB9A P51151 1/20 0.41
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7208461 1.00 MMP13 (1.00) MMP13MMP8MMP1ADAM17MMP2
SCHEMBL7208471 1.00 MMP13 (1.00) MMP13MMP8MMP1ADAM17MMP2
SCHEMBL7208473 1.00 MMP13 (1.00) MMP13MMP8MMP1ADAM17MMP2
SCHEMBL8438391 0.86 MMP13 (0.74) MMP13MMP8MMP1ADAM17MMP2
SCHEMBL27529540 0.81 MMP13 (0.68) MMP13MMP8MMP1MMP2MMP9
SCHEMBL1188309 0.79 MMP13 (0.73) MMP13MMP8MMP1ADAM17MMP2
SCHEMBL7212111 0.74 MMP13 (1.00) MMP13MMP8MMP1ADAM17MMP2
SCHEMBL10800122 0.73 MMP13 (0.58) MMP13MMP8MMP1MMP2MMP9
SCHEMBL30748417 0.73 MMP13 (0.60) MMP13MMP8MMP1MMP2MMP9
SCHEMBL6932129 0.72 MMP9 (0.59) MMP13MMP8MMP1ADAM17MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed