SCHEMBL7208669

SCHEMBL7208669

C=CC(Nc1ccc(NC(C=C)N2CCOC2)c2c1C(=O)c1ccccc1C2=O)N1CCOC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TERT O14746 3/20 0.43
MAPT P10636 5/20 0.39
L3MBTL1 Q9Y468 4/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TDP1 Q9NUW8 1/20 0.39
NSD2 O96028 4/20 0.37
LMNA P02545 2/20 0.37
APAF1 O14727 5/20 0.36
ALDH1A1 P00352 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
KDM4E B2RXH2 2/20 0.36
HTT P42858 1/20 0.36
TDP2 O95551 2/20 0.35
BLM P54132 2/20 0.35
GALK1 P51570 1/20 0.35
ATM Q13315 1/20 0.35
HKDC1 Q2TB90 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11213982 0.85 CYP19A1 (0.34) TERTMAPTL3MBTL1MEN1KMT2A
SCHEMBL6438245 0.68 MAOA (0.41) TERTMAPTL3MBTL1MEN1KMT2A
SCHEMBL7208670 0.68 TERT (0.46) TERTMAPTL3MBTL1MEN1KMT2A
SCHEMBL11187033 0.66 CYP19A1 (0.36) TERTMAPTL3MBTL1MEN1KMT2A
SCHEMBL1802818 0.65 MEN1 (0.42) TERTMAPTL3MBTL1MEN1KMT2A
SCHEMBL9239538 0.63 MALT1 (0.66) TERTMAPTL3MBTL1MEN1KMT2A
SCHEMBL7208666 0.62 NPC1 (0.39) TERTMAPTL3MBTL1MEN1KMT2A
SCHEMBL9239646 0.62 NQO1 (0.71) TERTMAPTMEN1KMT2ANPC1
SCHEMBL10622198 0.61 MEN1 (0.54) MAPTL3MBTL1MEN1KMT2ANPC1
SCHEMBL29351322 0.61 MEN1 (0.52) TERTMAPTL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0710689-B1 Polymeric antitumor agents WYETH CORP (US) 2003-05-02 EP disclosed
US-5609867-A POLYAMIDES FROM DIAMINE MONOMERS CONTAINING ANTHRAQUINONE, ANTHRAPYRAZOLE, AZA-ANTHRAQUINONE, AND DIAZA-ANTHRAQUINONE RINGS AMERICAN CYANAMID COMPANY (US) 1997-03-11 US disclosed
EP-0710689-A2 Polymeric antitumor agents American Cyanamid Company (US) 1996-05-08 EP disclosed
US-4715993-A FROM SALTS, USING AMMONIA OR METHYLAMINE AMERICAN CYANAMID COMPANY (US) 1987-12-29 US disclosed
US-4526788-A Polymeric[[(oxazolidinyl)alkyl]amino]anthraquinones AMERICAN CYANAMID COMPANY (US) 1985-07-02 US disclosed
US-4526788-A Polymeric[[(oxazolidinyl)alkyl]amino]anthraquinones AMERICAN CYANAMID COMPANY (US) 1985-07-02 US disclosed
EP-0122417-A2 Polymeric(((oxazolidinyl)alkyl)amino)anthraquinones AMERICAN CYANAMID COMPANY (US) 1984-10-24 EP disclosed