SCHEMBL7208834

SCHEMBL7208834

COc1ccc(Oc2c(Cl)cc([N+](=O)[O-])cc2Cl)cc1S(=O)(=O)Cl.COc1ccc(Oc2c(Cl)cc([N+](=O)[O-])cc2Cl)cc1S(=O)(=O)Cl

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE7A Q13946 1/20 0.42
MAPT P10636 5/20 0.42
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
HPGD P15428 3/20 0.42
ALDH1A1 P00352 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
CYP2C9 P11712 2/20 0.41
NPC1 O15118 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
GAA P10253 2/20 0.40
PKM P14618 1/20 0.40
TRPV4 Q9HBA0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4961573 1.00 PDE7A (0.42) PDE7AMAPTLMNASMN1; SMN2HPGD
SCHEMBL7039626 0.93 MEN1 (0.41) PDE7AMAPTLMNASMN1; SMN2HPGD
SCHEMBL6273901 0.89 ALDH1A1 (0.41) PDE7AMAPTLMNASMN1; SMN2HPGD
SCHEMBL6274128 0.88 MAPT (0.43) PDE7AMAPTLMNASMN1; SMN2HPGD
SCHEMBL14451769 0.85 ALDH1A1 (0.47) PDE7ALMNAALDH1A1POLBMEN1
SCHEMBL4963123 0.84 HSPB1 (0.41) PDE7AMAPTLMNASMN1; SMN2HPGD
SCHEMBL6660363 0.84 ALDH1A1 (0.57) LMNASMN1; SMN2HPGDALDH1A1RAB9A
SCHEMBL7042931 0.83 MEN1 (0.43) PDE7AMAPTLMNASMN1; SMN2HPGD
SCHEMBL4964933 0.82 CYP2C9 (0.43) PDE7AMAPTLMNASMN1; SMN2HPGD
SCHEMBL4961548 0.82 L3MBTL1 (0.52) SMN1; SMN2ALDH1A1NPSR1KMT2APKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268404-A1 MALONAMIC ACIDS AND DERIVATIVES THEREOF AS THYROID RECEPTOR LIGANDS Pfizer Products Inc. (US) 2003-01-02 EP disclosed
WO-2001072692-A1 MALONAMIC ACIDS AND DERIVATIVES THEREOF AS THYROID RECEPTOR LIGANDS PFIZER PRODUCTS INC. (US) 2001-10-04 WO disclosed