SCHEMBL7210290

SCHEMBL7210290

NS(=O)(=O)c1ccc(-n2cccc2-c2ccncc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.70
PTGS1 P23219 2/20 0.70
CA2 P00918 7/20 0.49
CA1 P00915 6/20 0.49
CA9 Q16790 6/20 0.49
CA12 O43570 4/20 0.49
ALDH1A1 P00352 1/20 0.45
CYP2C9 P11712 1/20 0.43
PDPK1 O15530 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215299 0.94 PTGS2 (0.70) PTGS2PTGS1CA2CA1CA9
SCHEMBL7212148 0.86 PTGS2 (0.76) PTGS2PTGS1CA2CA1CA9
SCHEMBL7210405 0.86 PTGS2 (0.63) PTGS2PTGS1CA2CA1CA9
SCHEMBL7211917 0.85 PTGS2 (0.70) PTGS2PTGS1CYP2C9
SCHEMBL7210655 0.83 PTGS2 (0.76) PTGS2PTGS1CA2CA1CA9
SCHEMBL7216312 0.83 PTGS2 (0.75) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL7216214 0.83 PTGS2 (0.75) PTGS2PTGS1CYP2C9PDPK1
SCHEMBL7211950 0.82 PTGS2 (0.74) PTGS2PTGS1CA2CA1CA9
SCHEMBL5308822 0.82 PTGS2 (0.74) PTGS2PTGS1CA2CA1CA9
SCHEMBL2463751 0.82 PTGS2 (1.00) PTGS2PTGS1CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP claimed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed