SCHEMBL7210405

SCHEMBL7210405

NS(=O)(=O)c1ccc(-n2cccc2-c2cccnc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.63
PTGS1 P23219 2/20 0.63
CA2 P00918 5/20 0.61
CA1 P00915 4/20 0.61
CA9 Q16790 4/20 0.61
CA12 O43570 2/20 0.61
CA4 P22748 1/20 0.50
CA7 P43166 1/20 0.50
ALDH1A1 P00352 1/20 0.48
CYP2A6 P11509 1/20 0.48
CYP2A13 Q16696 1/20 0.48
DYRK1A Q13627 1/20 0.46
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
KMT2A Q03164 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
FYN P06241 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7210775 0.86 PTGS2 (0.64) PTGS2PTGS1ALDH1A1CYP2A6CYP2A13
SCHEMBL7210290 0.86 PTGS2 (0.70) PTGS2PTGS1CA2CA1CA9
SCHEMBL7212148 0.84 PTGS2 (0.76) PTGS2PTGS1CA2CA1CA9
SCHEMBL7215299 0.83 PTGS2 (0.70) PTGS2PTGS1CA2CA1CA9
SCHEMBL7212078 0.82 PTGS2 (0.58) PTGS2PTGS1CA2CA1CA9
SCHEMBL7215905 0.79 PTGS2 (0.58) PTGS2PTGS1CA2CA1CA9
SCHEMBL8506129 0.78 CA2 (0.50) PTGS2PTGS1CA2CA1CA9
SCHEMBL7210655 0.78 PTGS2 (0.76) PTGS2PTGS1CA2CA1CA9
SCHEMBL10059589 0.77 CA2 (0.65) PTGS2CA2CA1CA9CA12
SCHEMBL5311727 0.77 PTGS2 (0.74) PTGS2PTGS1CA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP claimed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed