SCHEMBL7211797

SCHEMBL7211797

CC(C)(C)OC(=O)NCCCCCCNC(=O)c1c(Cl)ccc(N)c1O

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
TDP1 Q9NUW8 1/20 0.47
CA12 O43570 5/20 0.45
CA1 P00915 5/20 0.45
CA2 P00918 5/20 0.45
CA9 Q16790 5/20 0.45
DRD2 P14416 4/20 0.44
STK17B O94768 1/20 0.42
STK17A Q9UEE5 1/20 0.42
NPSR1 Q6W5P4 1/20 0.41
CSNK2A2 P19784 1/20 0.41
CSNK2A1 P68400 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7216748 0.82 ALDH1A1 (0.45) MAOAMAOBTDP1CA12CA1
SCHEMBL7217938 0.81 NAMPT (0.49) TDP1CA1CA2NPSR1
SCHEMBL7211897 0.78 CXCR2 (0.50) DRD2
SCHEMBL7212993 0.77 CXCR2 (0.54) TDP1CA12CA1CA2CA9
SCHEMBL7213015 0.76 ALDH1A1 (0.46) MAOAMAOBTDP1CA12CA1
SCHEMBL6563429 0.76 CXCR1 (0.45) MAOAMAOBTDP1CA12CA1
SCHEMBL22939550 0.74 TDP1 (0.55) MAOAMAOBTDP1CA12CA1
SCHEMBL3904926 0.74 TDP1 (0.55) MAOAMAOBTDP1CA12CA1
SCHEMBL6563501 0.74 CXCR2 (0.42) CA12CA1CA2CA9STK17B
SCHEMBL30448505 0.73 HDAC1 (0.48) MAOAMAOBTDP1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237548-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-07-23 EP disclosed
EP-1237548-A1 IL-8 RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-09-11 EP disclosed
WO-2001034141-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-17 WO disclosed