SCHEMBL7216748

SCHEMBL7216748

CC(C)(C)OC(=O)NCCCCCCNC(=O)c1c(Cl)ccc([N+](=O)[O-])c1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
TDP1 Q9NUW8 1/20 0.43
HSP90AA1 P07900 1/20 0.43
HPGD P15428 1/20 0.43
CA12 O43570 4/20 0.42
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
CA9 Q16790 4/20 0.42
DRD2 P14416 4/20 0.42
NPSR1 Q6W5P4 2/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
GPR55 Q9Y2T6 1/20 0.40
STK17B O94768 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7213015 0.90 ALDH1A1 (0.46) ALDH1A1TDP1HSP90AA1HPGDCA12
SCHEMBL7211797 0.82 MAOA (0.48) TDP1CA12CA1CA2CA9
SCHEMBL7212951 0.82 NAMPT (0.46) ALDH1A1HSP90AA1HPGDCA1CA2
SCHEMBL6564213 0.78 CXCR1 (0.42) ALDH1A1HSP90AA1HPGDCA12CA1
SCHEMBL6563381 0.76 MAPK1 (0.43) ALDH1A1HSP90AA1HPGDCA12CA1
SCHEMBL30448496 0.75 ALDH1A1 (0.51) ALDH1A1TDP1HSP90AA1HPGDCA12
SCHEMBL7656153 0.75 MMP2 (0.43) ALDH1A1CA12CA1CA2CA9
SCHEMBL7211897 0.74 CXCR2 (0.50) DRD2MAPT
SCHEMBL3911624 0.74 HDAC1 (0.60) ALDH1A1TDP1LMNAMAPT
SCHEMBL7212993 0.73 CXCR2 (0.54) TDP1CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1237548-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2003-07-23 EP disclosed
EP-1237548-A1 IL-8 RECEPTOR ANTAGONISTS SmithKline Beecham Corporation (US) 2002-09-11 EP disclosed
WO-2001034141-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-17 WO disclosed