SCHEMBL7212256

SCHEMBL7212256

COC(=O)[C@]1(O)CCCN1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.38
USP2 O75604 1/20 0.34
HSD11B1 P28845 1/20 0.33
CYP3A4 P08684 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33
CYP2C9 P11712 3/20 0.31
GAA P10253 2/20 0.31
CYP2C19 P33261 1/20 0.31
CYP2D6 P10635 2/20 0.31
MAPT P10636 2/20 0.31
HIF1A Q16665 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CASP6 P55212 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KCNH2 Q12809 1/20 0.31
CYP1A2 P05177 2/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6284592 0.79 OPRM1 (0.38) KDM4EKCNH2
SCHEMBL3665848 0.76 NPSR1 (0.35) NPSR1USP2CYP3A4MEN1KMT2A
SCHEMBL9762967 0.74
SCHEMBL845600 0.74
SCHEMBL845602 0.74
SCHEMBL10792890 0.73 ALDH1A1 (0.34) NPSR1USP2CYP3A4MEN1KMT2A
SCHEMBL6286104 0.72 ALDH1A1 (0.35) KDM4ELMNAALDH1A1
SCHEMBL4309286 0.71 GRIN2B (0.40) USP2
SCHEMBL4437296 0.71 GRIN2B (0.40) USP2
SCHEMBL692636 0.71 GRIN2B (0.40) USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102036966-A Difluorinated tripeptides as HCV serine protease inhibitors ENANTA PHARM INC 2011-04-27 CN disclosed
CN-101977621-A Fluorinated tripeptide hcv serine protease inhibitors ENANTA PHARM INC 2011-02-16 CN disclosed
US-6613738-B1 Comprising 1,2-dihydroxy-homotyrosine, 4-hydroxyproline, threonine, glutamine, 3-,4-dihydroxymethylproline, 4,5-dihydroxyornithine and lipid HMV CORPORATION 2003-09-02 US disclosed
WO-2000009735-A1 A CYCLIC LIPOPEPTIDE FROM CRYPTOSPORIOPSIS QUERCINA POSSESSING ANTIFUNGAL ACTIVITY STROBEL GARY A (US) 2000-02-24 WO disclosed