SCHEMBL7213313

SCHEMBL7213313

COc1cc(CC(=O)N[C@@H](CC(C)C)C(=O)NC[C@@H](C(=O)O)c2ccc3c(c2)OCO3)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 11/20 0.52
ITGA4 P13612 11/20 0.52
KMT2A Q03164 2/20 0.47
P2RX7 Q99572 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
TP53 P04637 1/20 0.41
CTSD P07339 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7467442 0.93 KMT2A (0.49) ITGB1ITGA4KMT2ANPC1CTSD
SCHEMBL7219807 0.89 ITGB1 (0.54) ITGB1ITGA4NPC1RAB9A
SCHEMBL7459141 0.84 NPC1 (0.41) ITGB1ITGA4KMT2ANPC1RAB9A
SCHEMBL7464392 0.84 NPC1 (0.41) ITGB1ITGA4KMT2ANPC1RAB9A
SCHEMBL7468356 0.84 KMT2A (0.45) ITGB1ITGA4KMT2ARAB9A
SCHEMBL7461109 0.83 KMT2A (0.45) ITGB1ITGA4KMT2ARAB9ATP53
SCHEMBL7467339 0.83 KMT2A (0.45) ITGB1ITGA4KMT2ARAB9ATP53
SCHEMBL7464096 0.83 NPC1 (0.43) ITGB1ITGA4KMT2AP2RX7NPC1
SCHEMBL7462350 0.83 NPC1 (0.43) ITGB1ITGA4KMT2AP2RX7NPC1
SCHEMBL7462016 0.82 KMT2A (0.49) ITGB1ITGA4KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6624152-B2 Inhibition and prevention of cell adhesion and cell adhesion-mediated pathologies. This invention relates to pharmaceutical formulations comprising these compounds and methods of using them for inflammatory and autoimmune diseases BIOGEN, INC. 2003-09-23 US claimed
EP-0805796-B1 CELL ADHESION INHIBITORS BIOGEN INC (US) 2002-12-11 EP claimed