SCHEMBL7214904

SCHEMBL7214904

CCOC(=O)c1cccc(-c2nc(-c3ccc(Cl)cc3)cs2)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.61
KDM4E B2RXH2 2/20 0.53
MEN1 O00255 1/20 0.53
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
KMT2A Q03164 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
SREBF2 Q12772 1/20 0.50
EIF4E P06730 1/20 0.49
LMNA P02545 2/20 0.49
MAPT P10636 2/20 0.49
ATM Q13315 1/20 0.49
TSHR P16473 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
TRPM8 Q7Z2W7 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1505172 0.89 L3MBTL1 (0.54) L3MBTL1KDM4EMEN1NPC1RAB9A
SCHEMBL7220970 0.88 CDC25A (0.60) L3MBTL1MEN1NPC1RAB9AKMT2A
SCHEMBL7221010 0.88 L3MBTL1 (0.54) L3MBTL1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL7217168 0.87 KDM4E (0.66) L3MBTL1KDM4EMEN1NPC1RAB9A
SCHEMBL16180612 0.87 SMN1; SMN2 (0.59) L3MBTL1KDM4EMEN1NPC1RAB9A
SCHEMBL7215066 0.87 L3MBTL1 (0.52) L3MBTL1KDM4EMEN1NPC1RAB9A
SCHEMBL3824273 0.86 KDM4E (0.52) L3MBTL1KDM4EMEN1NPC1RAB9A
SCHEMBL23742629 0.85 KDM4E (0.52) L3MBTL1KDM4EMEN1NPC1RAB9A
SCHEMBL23742625 0.85 TRPM8 (0.57) L3MBTL1KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL7221374 0.83 L3MBTL1 (0.55) L3MBTL1KDM4ESMN1; SMN2EIF4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545009-B1 Imidazole, oxazole and thiazole derivatives for regulation of peroxisome proliferator-activated receptor function; improving insulin resistance, treating impaired glucose tolerance and obesity, enhancing insulin sensitivity, etc. TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-04-08 US disclosed
CN-1314899-A Retinoid-associated receptor regulators TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-09-26 CN disclosed
EP-1092711-A1 RETINOID-ASSOCIATED RECEPTOR REGULATORS Takeda Chemical Industries, Ltd. (JP) 2001-04-18 EP disclosed