SCHEMBL7215217

SCHEMBL7215217

COC(=O)c1ccc(-c2nc(-c3ccc(Br)cc3)cs2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.59
RAB9A P51151 6/20 0.59
SMN1; SMN2 Q16637 6/20 0.59
NPC1 O15118 5/20 0.59
ALDH1A1 P00352 4/20 0.59
LMNA P02545 2/20 0.58
MAPT P10636 7/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
SIRT5 Q9NXA8 1/20 0.53
MEN1 O00255 6/20 0.52
KMT2A Q03164 6/20 0.52
CYP19A1 P11511 1/20 0.52
POLB P06746 1/20 0.50
ATM Q13315 1/20 0.50
GAA P10253 1/20 0.49
NPSR1 Q6W5P4 1/20 0.47
HPGD P15428 1/20 0.46
GRM1 Q13255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7215145 0.88 MAPT (0.61) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL7217216 0.86 RAB9A (0.71) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
Bromide SCHEMBL7215820 0.86 KDM4E (0.59) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL5698744 0.86 KDM4E (0.59) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL7217201 0.84 KDM4E (0.56) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL7221977 0.84 RAB9A (0.56) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL27560241 0.84 LOXL2 (0.61) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL7221406 0.83 MAPT (0.59) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL13779213 0.83 MAPT (0.54) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL7221752 0.83 KDM4E (0.78) KDM4ERAB9ASMN1; SMN2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545009-B1 Imidazole, oxazole and thiazole derivatives for regulation of peroxisome proliferator-activated receptor function; improving insulin resistance, treating impaired glucose tolerance and obesity, enhancing insulin sensitivity, etc. TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-04-08 US disclosed
CN-1314899-A Retinoid-associated receptor regulators TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-09-26 CN disclosed
EP-1092711-A1 RETINOID-ASSOCIATED RECEPTOR REGULATORS Takeda Chemical Industries, Ltd. (JP) 2001-04-18 EP disclosed