SCHEMBL7215974

SCHEMBL7215974

NS(=O)(=O)c1ccc(-c2cccn2C2CCCCC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.55
CA2 P00918 16/20 0.51
CA9 Q16790 14/20 0.51
CA1 P00915 14/20 0.51
CA12 O43570 13/20 0.51
PTGS1 P23219 1/20 0.47
CA7 P43166 2/20 0.43
CA5A P35218 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
CA4 P22748 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8250269 0.78 SLC18A3 (0.43) CA2CA9CA1CA12
SCHEMBL28601412 0.77 CA12 (0.39) PTGS2CA2CA9CA1CA12
SCHEMBL28598700 0.77 GLA (0.41) PTGS2CA2CA9CA1CA12
SCHEMBL8505690 0.76 PTGES2 (0.37) PTGS2CA2CA9CA1CA12
SCHEMBL12504926 0.75 GLA (0.39) PTGS2CA2CA9CA1CA12
SCHEMBL28602234 0.74 ALDH1A1 (0.46) CA2CA9CA1CA12
SCHEMBL28601637 0.74 SMN1; SMN2 (0.43)
SCHEMBL28606349 0.74 KCNH2 (0.44)
SCHEMBL7209882 0.73 PTGS2 (0.78) PTGS2CA2CA9CA1CA12
SCHEMBL28609103 0.71 PGR (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP claimed
EP-0946507-B1 SUBSTITUTED PYRROLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2003-09-24 EP claimed
EP-1369415-A1 Substituted pyrrolyl compounds for the treatment of inflammation G.D. SEARLE & CO. (US) 2003-12-10 EP disclosed