SCHEMBL7216530

SCHEMBL7216530

COC(=O)C1CCCc2ccc(OCc3ccc(-c4ccccc4)cc3)cc2C1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.51
MAOB P27338 6/20 0.51
GSTP1 P09211 1/20 0.45
RXRA P19793 3/20 0.43
RXRB P28702 3/20 0.43
RXRG P48443 3/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ADAMTS4 O75173 1/20 0.43
MMP2 P08253 1/20 0.43
MMP13 P45452 1/20 0.43
MMP14 P50281 1/20 0.43
ADAMTS5 Q9UNA0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223230 0.94 MAOA (0.58) MAOAMAOBRXRARXRBRXRG
SCHEMBL7216956 0.89 MAOB (0.60) MAOAMAOBRXRARXRBRXRG
SCHEMBL7222116 0.80 ACHE (0.49) MAPTKDM4E
SCHEMBL7755671 0.79 FAAH (0.43)
SCHEMBL9621233 0.78 NPC1 (0.46) NPC1RAB9A
SCHEMBL7218099 0.77 MAOB (0.82) MAOAMAOBGSTP1NPC1RAB9A
SCHEMBL2166539 0.74 NPC1 (0.44) MAOAMAOBNPC1RAB9AMAPT
SCHEMBL9621088 0.74 NPC1 (0.43) NPC1RAB9ASMPD1
SCHEMBL4875547 0.73 SMN1; SMN2 (0.43) MAOAMAOBNPC1RAB9AMAPT
SCHEMBL14059398 0.73 TDP1 (0.38) MAPTKDM4EALDH1A1HPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627651-B1 Exhibiting preventive and therapeutic effects against HIV infectious diseases wherein R1 is an optionally substituted five- or six-membered ring group; X1 is a free valency or the like; W is a divalent group and inhibitors of HIV (human TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1182195-A1 CYCLIC COMPOUNDS AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-27 EP disclosed