SCHEMBL7216573

SCHEMBL7216573

CCOC(=O)CN[C@@H](C(=O)O)C1CCCCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.43
TSHR P16473 2/20 0.42
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
THRB P10828 1/20 0.40
ATM Q13315 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
CYP2D6 P10635 1/20 0.39
MGAM O43451 1/20 0.37
GAA P10253 1/20 0.37
SI P14410 1/20 0.37
MGAM2 Q2M2H8 1/20 0.37
TP53 P04637 1/20 0.37
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP7 P09237 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7218526 0.98 F2 (0.43) F2TSHRALDH1A1NPSR1L3MBTL1
SCHEMBL8236141 0.80 L3MBTL1 (0.50) F2TSHRALDH1A1L3MBTL1KDM4E
SCHEMBL21468160 0.79 SMN1; SMN2 (0.41) TSHRALDH1A1KDM4EMMP1MMP2
SCHEMBL27733842 0.79 SMN1; SMN2 (0.41) TSHRALDH1A1KDM4EMMP1MMP2
SCHEMBL1410684 0.79 SMN1; SMN2 (0.41) TSHRALDH1A1KDM4EMMP1MMP2
SCHEMBL8991906 0.79 ALDH1A1 (0.42) F2ALDH1A1KDM4EMMP1MMP2
SCHEMBL6436784 0.78 TSHR (0.44) TSHRALDH1A1NPSR1L3MBTL1THRB
SCHEMBL14263864 0.78 TSHR (0.44) TSHRALDH1A1NPSR1L3MBTL1THRB
SCHEMBL6436779 0.78 TSHR (0.44) TSHRALDH1A1NPSR1L3MBTL1THRB
SCHEMBL7433429 0.77 ALDH1A1 (0.40) F2TSHRALDH1A1NPSR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6518434-B2 N-carboxyanhydrides (NCAs) are copupled directly to cyclic amino acids amide derivatives to form peptide linkage ASTRAZENECA AB (SE) 2003-02-11 US disclosed
EP-1257533-A1 NEW COUPLING PROCESS AstraZeneca AB (SE) 2002-11-20 EP disclosed
US-20020128452-A1 N-carboxyanhydrides (NCAs) are copupled directly to cyclic amino acids amide derivatives to form peptide linkage ASTRAZENECA AB (SE) 2002-09-12 US disclosed
WO-2001056986-A1 NEW COUPLING PROCESS ASTRAZENECA AB (SE) 2001-08-09 WO disclosed