SCHEMBL7217113

SCHEMBL7217113

COCC(N)CC(N)Cc1ccc(OC)c(OC)c1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.51
ALOX15 P16050 1/20 0.51
ALOX12 P18054 1/20 0.51
SIGMAR1 Q99720 8/20 0.50
CA2 P00918 1/20 0.50
KDM4E B2RXH2 1/20 0.49
ATM Q13315 1/20 0.49
STAT3 P40763 1/20 0.46
CYP19A1 P11511 1/20 0.46
AOC3 Q16853 1/20 0.44
ALDH1A1 P00352 1/20 0.44
PPARG P37231 1/20 0.44
PPARD Q03181 1/20 0.44
PPARA Q07869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16930335 0.85 SIGMAR1 (0.56) LDHAALOX15ALOX12SIGMAR1CA2
SCHEMBL17709282 0.82 SIGMAR1 (0.56) SIGMAR1
SCHEMBL2404037 0.81 LDHA (0.56) LDHAALOX15ALOX12SIGMAR1CA2
SCHEMBL10437147 0.81 KDM4E (0.58) LDHAALOX15ALOX12SIGMAR1CA2
SCHEMBL10842397 0.81 LDHA (0.56) LDHAALOX15ALOX12SIGMAR1CA2
SCHEMBL13623723 0.81 SIGMAR1 (0.47) ALOX15ALOX12SIGMAR1
SCHEMBL10776070 0.80 LDHA (0.58) LDHAALOX15ALOX12SIGMAR1CA2
SCHEMBL7290411 0.80 LDHA (0.58) LDHAALOX15ALOX12SIGMAR1CA2
SCHEMBL7298435 0.80 LDHA (0.58) LDHAALOX15ALOX12SIGMAR1CA2
Phyllanthin SCHEMBL503799 0.80 LDHA (0.57) LDHAALOX15ALOX12CA2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339702-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEK INHIBITORS WARNER-LAMBERT COMPANY (US) 2003-09-03 EP disclosed
WO-2001068619-A1 5-AMIDE SUBSTITUTED DIARYLAMINES AS MEX INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-09-20 WO disclosed