SCHEMBL7217150

SCHEMBL7217150

O=C(O)c1ccc(-c2nc(-c3ccc(OC(F)F)cc3)co2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP3 O14638 2/20 0.48
ENPP1 P22413 2/20 0.48
CHEK1 O14757 1/20 0.42
ALOX15 P16050 1/20 0.41
GFER P55789 1/20 0.41
ADAM17 P78536 1/20 0.41
KMT2A Q03164 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
SMO Q99835 2/20 0.40
ATM Q13315 1/20 0.40
PPARD Q03181 1/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EIF4E P06730 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12796882 0.87 MRGPRX4 (0.48) ENPP3ENPP1NR1H4SMONPC1
SCHEMBL7217142 0.86 ENPP3 (0.48) ENPP3ENPP1ALOX15GFERADAM17
SCHEMBL13287537 0.85 ENPP3 (0.49) ENPP3ENPP1CHEK1KMT2ANR1H4
SCHEMBL7215190 0.83 ENPP3 (0.70) ENPP3ENPP1CHEK1GFERKMT2A
SCHEMBL16378628 0.83 ENPP3 (0.70) ENPP3ENPP1CHEK1GFERKMT2A
SCHEMBL7215644 0.81 NPC1 (0.58) ENPP3ENPP1CHEK1KMT2ANR1H4
SCHEMBL7215456 0.81 NPC1 (0.58) ENPP3ENPP1CHEK1KMT2ANR1H4
SCHEMBL12243297 0.80 PLA2G4B (0.52) ENPP3ENPP1CHEK1NR1H4ALDH1A1
SCHEMBL16199783 0.79 HSD17B1 (0.57) ENPP3ENPP1CHEK1KMT2ASMO
SCHEMBL7221671 0.78 NPC1 (0.54) ENPP3ENPP1ALOX15KMT2ASMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6545009-B1 Imidazole, oxazole and thiazole derivatives for regulation of peroxisome proliferator-activated receptor function; improving insulin resistance, treating impaired glucose tolerance and obesity, enhancing insulin sensitivity, etc. TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-04-08 US disclosed
EP-1092711-A1 RETINOID-ASSOCIATED RECEPTOR REGULATORS Takeda Chemical Industries, Ltd. (JP) 2001-04-18 EP disclosed