SCHEMBL7217419

SCHEMBL7217419

CCC(CN)(c1ccccc1)c1cccc2ccccc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.41
TAAR1 Q96RJ0 1/20 0.39
HSD17B10 Q99714 3/20 0.35
HPGD P15428 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HIF1A Q16665 1/20 0.35
ACP3 P15309 1/20 0.34
ALDH1A1 P00352 3/20 0.33
TSHR P16473 3/20 0.33
CYP3A4 P08684 2/20 0.33
HTR1B P28222 2/20 0.33
KEAP1 Q14145 1/20 0.33
CA12 O43570 1/20 0.33
CA3 P07451 1/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8804043 0.84 KIF11 (0.38) KIF11HSD17B10HPGDCYP2C19CYP1A2
SCHEMBL27684804 0.84 KIF11 (0.41) KIF11TAAR1HSD17B10HPGDCYP2C19
SCHEMBL27684715 0.81 KIF11 (0.39) KIF11TAAR1HSD17B10HPGDCYP2C19
SCHEMBL2086206 0.78 TAAR1 (0.54) KIF11TAAR1CYP1A2CYP2D6CYP3A4
SCHEMBL28369183 0.76 ALDH1A1 (0.38) KIF11HSD17B10HPGDCYP2C19CYP1A2
SCHEMBL5010143 0.76 KIF11 (0.41) KIF11HSD17B10HPGDCYP2C19CYP1A2
SCHEMBL16721031 0.73 CYP2C19 (0.44) KIF11HSD17B10HPGDCYP2C19CYP1A2
SCHEMBL27684720 0.73 KIF11 (0.43) KIF11TAAR1HSD17B10HPGDCYP2C19
SCHEMBL9179221 0.73 KIF11 (0.46) KIF11TAAR1HSD17B10HPGDCYP2C19
SCHEMBL28039335 0.73 ALDH1A1 (0.35) KIF11HSD17B10HPGDCYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1148876-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2003-07-23 EP disclosed
EP-1070048-A4 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2001-11-07 EP disclosed
EP-1148876-A1 CALCILYTIC COMPOUNDS SmithKline Beecham Corporation (US) 2001-10-31 EP disclosed
EP-1070048-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2001-01-24 EP disclosed
WO-2000045816-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (GB) 2000-08-10 WO disclosed
WO-1999051569-A1 CALCILYTIC COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1999-10-14 WO disclosed