SCHEMBL7218189

SCHEMBL7218189

c1ccc(CN2CCC(NCc3ccc(-c4ccccc4)cc3)CC2)cc1

nearest known ligand 0.85

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 14/20 0.85
BACE1 P56817 14/20 0.85
BCHE P06276 11/20 0.85
MEN1 O00255 3/20 0.79
KMT2A Q03164 3/20 0.79
HTR5A P47898 2/20 0.79
HRH3 Q9Y5N1 1/20 0.68
RAB9A P51151 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14367985 0.92 ACHE (1.00) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL7695906 0.92 ACHE (0.92) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL7695958 0.89 HTR5A (0.77) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL7696728 0.88 ACHE (0.71) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL7696604 0.88 ACHE (0.71) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL7690757 0.88 ACHE (0.71) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL1803081 0.88 ACHE (1.00) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL16055288 0.87 ACHE (0.85) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL20492760 0.87 ACHE (1.00) ACHEBACE1BCHEMEN1KMT2A
SCHEMBL4205093 0.87 ACHE (1.00) ACHEBACE1BCHEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1322612-A1 SUBSTITUTED AMINO-AZA-CYCLOALKANES USEFUL AGAINST MALARIA Actelion Pharmaceuticals Ltd. (CH) 2003-07-02 EP disclosed
WO-2002024649-A1 SUBSTITUTED AMINO-AZA-CYCLOALKANES USEFUL AGAINST MALARIA ACTELION PHARMACEUTICALS LTD (CH) 2002-03-28 WO disclosed