SCHEMBL7218455

SCHEMBL7218455

COc1cccc2c1OC(CN1CC=C(c3c[nH]c4ncccc34)CC1)CO2.COc1cccc2c1O[C@H](Cc1cc(C)ccc1S(=O)(=O)O)CO2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 16/20 0.48
SLC6A4 P31645 8/20 0.48
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
PLK4 O00444 1/20 0.39
CHEK1 O14757 1/20 0.39
AURKA O14965 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
CHEK2 O96017 1/20 0.39
PRKCG P05129 1/20 0.39
CDK1 P06493 1/20 0.39
RET P07949 1/20 0.39
PIM1 P11309 1/20 0.39
FGFR1 P11362 1/20 0.39
PRKACA P17612 1/20 0.39
RPS6KB1 P23443 1/20 0.39
CDK2 P24941 1/20 0.39
MARK3 P27448 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5846334 0.88 HTR1A (0.53) HTR1ASLC6A4ADRA1DADRA1AADRA1B
SCHEMBL7215975 0.88 HTR1A (0.60) HTR1ASLC6A4
SCHEMBL5844134 0.87 HTR1A (0.61) HTR1ASLC6A4ADRA1DADRA1AADRA1B
SCHEMBL5845602 0.78 HTR1A (0.52) HTR1ASLC6A4
SCHEMBL5845943 0.78 ADRA1D (0.44) HTR1ASLC6A4ADRA1DADRA1AADRA1B
SCHEMBL5845948 0.78 ADRA1D (0.44) HTR1ASLC6A4ADRA1DADRA1AADRA1B
SCHEMBL7030051 0.78 HTR1A (0.61) HTR1ASLC6A4
SCHEMBL7034836 0.77 HTR1A (0.49) HTR1ASLC6A4
SCHEMBL7004959 0.76 HTR1A (0.54) HTR1ASLC6A4ADRA1DADRA1AADRA1B
SCHEMBL7034985 0.76 HTR1A (0.53) HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6559169-B2 For therapy of depression, anxiety, panic disorder, post-traumatic stress disorder, premenstrual dysphoric disorder attention deficit disorder,obsessive compulsive disorder, obesity, eating disorders, sexual dysfunction WYETH 2003-05-06 US disclosed