SCHEMBL5845602

SCHEMBL5845602

COc1ccc2c(c1)OC(CN1CC=C(c3c[nH]c4ccccc34)CC1)CO2.COc1ccc2c(c1)O[C@H](Cc1cc(C)ccc1S(=O)(=O)O)CO2

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 14/20 0.52
SLC6A4 P31645 1/20 0.52
DRD2 P14416 9/20 0.46
HTR2A P28223 3/20 0.46
DRD1 P21728 1/20 0.45
DRD3 P35462 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5845471 0.87 HTR1A (0.63) HTR1ASLC6A4DRD2HTR2ADRD1
SCHEMBL7030051 0.84 HTR1A (0.61) HTR1ASLC6A4DRD2HTR2A
SCHEMBL5846334 0.82 HTR1A (0.53) HTR1ASLC6A4DRD2HTR2A
SCHEMBL7215975 0.82 HTR1A (0.60) HTR1ASLC6A4DRD2
SCHEMBL7199693 0.78 MTNR1A (0.50)
SCHEMBL7218455 0.78 HTR1A (0.48) HTR1ASLC6A4
SCHEMBL7034985 0.77 HTR1A (0.53) HTR1ASLC6A4DRD2HTR2ADRD3
SCHEMBL7004959 0.77 HTR1A (0.54) HTR1ASLC6A4DRD2HTR2A
SCHEMBL7148718 0.77 HTR1A (0.52) HTR1ASLC6A4DRD2HTR2A
SCHEMBL7032693 0.76 HTR1A (0.51) HTR1ASLC6A4DRD2HTR2ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7041683-B2 Antidepressant azaheterocyclylmethyl derivatives of 2,3-dihydro-1, 4-benzodiozan WYETH (US) 2006-05-09 US disclosed
US-6559169-B2 For therapy of depression, anxiety, panic disorder, post-traumatic stress disorder, premenstrual dysphoric disorder attention deficit disorder,obsessive compulsive disorder, obesity, eating disorders, sexual dysfunction WYETH 2003-05-06 US disclosed