SCHEMBL7219598

SCHEMBL7219598

CN(C)C(=O)c1c(C(C)(C)C)cc(C(C)(C)C)cc1C(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLRA3 O75311 1/20 0.39
GLRB P48167 1/20 0.39
NR1H4 Q96RI1 2/20 0.38
EPHX2 P34913 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB2 P47870 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP2C19 P33261 1/20 0.37
LMNA P02545 2/20 0.37
RECQL P46063 1/20 0.37
NR5A2 O00482 1/20 0.36
NR5A1 Q13285 1/20 0.36
RXRA P19793 2/20 0.35
RXRB P28702 1/20 0.35
RXRG P48443 1/20 0.35
GABBR2 O75899 1/20 0.35
GABBR1 Q9UBS5 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30773074 0.80 NR5A2 (0.51) GLRA3GLRBGABRA1GABRB2HTT
SCHEMBL14825538 0.78 GLRA3 (0.42) GLRA3GLRBGABRA1GABRB2KMT2A
SCHEMBL6466602 0.78 GLRA3 (0.57) GLRA3GLRBGABRA1GABRB2CYP2C19
SCHEMBL14988234 0.77 GLRA3 (0.41) GLRA3GLRBNR1H4EPHX2GABRA1
SCHEMBL28419884 0.77 GLRA3 (0.55) GLRA3GLRBGABRA1GABRB2CYP2C19
SCHEMBL5997582 0.75 GLRA3 (0.36) GLRA3GLRBGABRA1GABRB2CYP2C19
SCHEMBL7217663 0.73 KMT2A (0.55) NR1H4KMT2AALDH1A1HSP90AA1NPC1
SCHEMBL7225441 0.73 NR5A2 (0.42) GLRA3GLRBNR1H4EPHX2GABRA1
SCHEMBL7218380 0.73 TP53 (0.41) HTTNR5A2NR5A1ALDH1A1RAB9A
SCHEMBL16147679 0.72 GLRA3 (0.55) GLRA3GLRBGABRA1GABRB2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6521603-B2 Amide, thioamide, amidine and thioester derivatives containing a benzene, pyridine, thiophene, furan, pyrrole, pyrazole, thiazole or isothiazole ring MONSANTO TECHNOLOGY LLC 2003-02-18 US claimed