SCHEMBL7219639

SCHEMBL7219639

NC(c1ccccc1)(c1ccccc1)C1CCN(CCCN2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.55
DRD2 P14416 2/20 0.54
ALDH1A1 P00352 1/20 0.53
DRD3 P35462 2/20 0.51
MAOB P27338 1/20 0.51
HTR7 P34969 1/20 0.51
HRH1 P35367 1/20 0.51
HTR2B P41595 1/20 0.51
ACHE P22303 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9253176 0.85 HRH1 (0.60) HTR1ADRD2ALDH1A1HRH1
SCHEMBL5729030 0.82 HRH1 (0.62) HTR1ADRD2HRH1
SCHEMBL29459507 0.78 HTR1A (0.62) HTR1ADRD2ALDH1A1DRD3MAOB
SCHEMBL26992312 0.78 HTR1A (0.62) HTR1ADRD2ALDH1A1DRD3MAOB
SCHEMBL13469510 0.78 HTR1A (0.79) HTR1ADRD2DRD3MAOB
SCHEMBL7989673 0.78 HTR1A (0.62) HTR1ADRD2ALDH1A1DRD3MAOB
SCHEMBL5113354 0.77 HTR1A (0.61) HTR1ADRD2ALDH1A1DRD3MAOB
SCHEMBL10479167 0.77 HRH1 (0.58) HRH1
SCHEMBL13590304 0.76 HTR1A (0.53) HTR1ADRD2ALDH1A1DRD3HTR7
SCHEMBL5425845 0.76 HTR1A (0.53) HTR1ADRD2ALDH1A1DRD3HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6627630-B1 Preventing or treating allergic skin diseases such as contact dermatitis, pruritus, dried dermatitis, acute urticaria prurigo and antiallergins TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-09-30 US disclosed
EP-1243271-A1 NASAL DROPS CONTAINING FUSED PYRIDAZINE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2002-09-25 EP disclosed
US-6248740-B1 FOR SUPPRESSION OF HISTAMINE OR EOSINOPHIL CHEMOTAXIS TO TREAT ASTHMA; ANTIALLERGENIC TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-06-19 US disclosed