SCHEMBL7219981

SCHEMBL7219981

N#Cc1c(-c2ccccc2)ccnc1-c1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
L3MBTL1 Q9Y468 2/20 0.61
CYP1A2 P05177 1/20 0.61
CYP2C9 P11712 1/20 0.61
CYP2C19 P33261 1/20 0.61
NPC1 O15118 1/20 0.54
MAPT P10636 1/20 0.54
CRHBP P24387 1/20 0.54
RAB9A P51151 1/20 0.54
CRHR2 Q13324 1/20 0.54
KDM4E B2RXH2 2/20 0.52
LMNA P02545 1/20 0.52
ADORA1 P30542 8/20 0.49
ADORA2A P29274 6/20 0.49
LRRK2 Q5S007 1/20 0.46
SQOR Q9Y6N5 1/20 0.44
CCNA2 P20248 1/20 0.44
CDK2 P24941 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27544440 0.81 ALDH1A1 (0.61) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2
SCHEMBL3089786 0.81 ADORA2A (0.56) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2
SCHEMBL3089781 0.81 ADORA2A (0.56) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2
SCHEMBL5329331 0.80 ADORA1 (0.56) ADORA1ADORA2ACDK2HSD17B10
SCHEMBL17971409 0.80 ALDH1A1 (0.59) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2
SCHEMBL16681058 0.80 ALDH1A1 (0.59) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2
SCHEMBL3205196 0.80 ALDH1A1 (0.59) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2
SCHEMBL12612051 0.78
SCHEMBL2977679 0.76 ALDH1A1 (0.44) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2
SCHEMBL2977681 0.76 ALDH1A1 (0.55) ALDH1A1MEN1KMT2AL3MBTL1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020146636-A1 COMPOUNDS AND METHODS FOR TREATING OR PREVENTING HEART FAILURE DREXEL UNIVERSITY (US) 2020-07-16 WO disclosed
US-6603007-B1 Intermediates in the fields of pharmaceuticals, agrichemicals, ligands, silver halide photosensitive materials, liquid crystals, surfactants, electrophotography and organic electroluminescence SANKIO CHEMICAL CO., LTD. (JP) 2003-08-05 US disclosed
EP-1231207-A1 NOVEL BIPYRIDYL DERIVATIVES Sankio Chemical Co., Ltd. (JP) 2002-08-14 EP disclosed